SCHEMBL28622161

SCHEMBL28622161

CN(C/C=C/C#CC(C)(C)C)C(=O)c1cccc2ccccc12

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.59
LMNA P02545 2/20 0.59
CYP2D6 P10635 2/20 0.59
ADRA2A P08913 1/20 0.59
SLC6A2 P23975 1/20 0.59
SQLE Q14534 1/20 0.59
PLK1 P53350 1/20 0.40
MMP3 P08254 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
NR4A1 P22736 1/20 0.37
NR4A2 P43354 1/20 0.37
NR4A3 Q92570 1/20 0.37
CNR1 P21554 1/20 0.37
CNR2 P34972 1/20 0.37
PTPN1 P18031 1/20 0.37
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
GMNN O75496 1/20 0.36
ALDH1A1 P00352 1/20 0.36
TP53 P04637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL30855369 0.99 SIGMAR1 (0.58) SIGMAR1LMNACYP2D6ADRA2ASLC6A2
SCHEMBL28616636 0.79 NR1I2 (0.54) SIGMAR1LMNACYP2D6SLC6A2PLK1
SCHEMBL28616637 0.79 NR1I2 (0.54) SIGMAR1LMNACYP2D6SLC6A2PLK1
SCHEMBL21591961 0.76 SIGMAR1 (0.65) SIGMAR1LMNACYP2D6ADRA2ASLC6A2
Terbinafine SCHEMBL1178093 0.76 CYP2D6 (0.87) SIGMAR1LMNACYP2D6ADRA2ASLC6A2
Terbinafine SCHEMBL2793602 0.76 CYP2D6 (0.87) SIGMAR1LMNACYP2D6ADRA2ASLC6A2
Hydrochloric Acid SCHEMBL30408182 0.75 SIGMAR1 (0.64) SIGMAR1LMNACYP2D6ADRA2ASLC6A2
Hydrochloric Acid SCHEMBL31374682 0.75 SIGMAR1 (0.64) SIGMAR1LMNACYP2D6ADRA2ASLC6A2
Terbinafine SCHEMBL2821945 0.75 CYP2D6 (0.85) SIGMAR1LMNACYP2D6ADRA2ASLC6A2
SCHEMBL3254626 0.74 SQLE (0.69) SIGMAR1LMNACYP2D6ADRA2ASLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113277963-B Amine compound and preparation method and application thereof 南京工业大学 2022-11-04 CN disclosed
CN-113277963-A Amine compound and preparation method and application thereof 南京工业大学 2021-08-20 CN disclosed