SCHEMBL28624866

SCHEMBL28624866

CCOC(=O)C1=NC=CC=CO1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.39
TSHR P16473 1/20 0.38
KDM4E B2RXH2 4/20 0.36
ALDH1A1 P00352 3/20 0.36
POLB P06746 2/20 0.36
PKM P14618 1/20 0.36
CA12 O43570 3/20 0.36
CA1 P00915 3/20 0.36
CA2 P00918 3/20 0.36
CA7 P43166 3/20 0.36
CA9 Q16790 3/20 0.36
CA14 Q9ULX7 3/20 0.36
ESR1 P03372 1/20 0.36
ESR2 Q92731 1/20 0.36
NR1H2 P55055 1/20 0.35
NR1H3 Q13133 1/20 0.35
LMNA P02545 1/20 0.35
CYP3A4 P08684 1/20 0.35
MAOA P21397 1/20 0.35
CYP2C9 P11712 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4919337 0.70 TSHR (0.41) CYP1A2TSHRKDM4EALDH1A1POLB
SCHEMBL28364501 0.67 CYP1A2 (0.39) CYP1A2TSHRKDM4EALDH1A1POLB
SCHEMBL29210425 0.66 TSHR (0.48) CYP1A2TSHRALDH1A1CA12CA1
SCHEMBL3677772 0.64
SCHEMBL30569264 0.63 CYP1A2 (0.39) CYP1A2TSHRKDM4EALDH1A1CA12
SCHEMBL28347204 0.63
SCHEMBL1427719 0.62 CYP1A2 (0.44) CYP1A2TSHRKDM4EALDH1A1CA12
SCHEMBL19102899 0.60 CYP1A2 (0.46) CYP1A2TSHRKDM4EALDH1A1POLB
SCHEMBL27821848 0.60 HCAR2 (0.52) CYP1A2TSHRALDH1A1CA12CA1
SCHEMBL362159 0.60 TSHR (0.63) CYP1A2TSHRKDM4EALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115867557-A Azepine fused ring compounds and medical application thereof 中国医药研究开发中心有限公司 2023-03-28 CN disclosed
CN-112689636-A Novel heteroatom aromatic amide derivative and drug containing the same 科研制药株式会社 2021-04-20 CN disclosed