SCHEMBL286274

SCHEMBL286274

O=C(O)c1cc(OCc2conc2-c2ccc(F)cn2)n[nH]1

nearest known ligand 0.51

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GABRA5 P31644 19/20 0.51
CA12 O43570 1/20 0.39
ALPL P05186 1/20 0.39
RPA1 P27694 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL286362 0.89 GABRA5 (0.48) GABRA5ALPL
SCHEMBL285835 0.83 GABRA5 (0.43) GABRA5
SCHEMBL1779461 0.81 GABRA5 (0.52) GABRA5
SCHEMBL2926043 0.80 GABRA5 (0.65) GABRA5
SCHEMBL286487 0.80 GABRA5 (0.68) GABRA5
SCHEMBL27865421 0.74 GABRA5 (0.55) GABRA5
SCHEMBL2933362 0.73 GABRA5 (0.68) GABRA5
SCHEMBL1776175 0.73 GABRA5 (0.48) GABRA5
SCHEMBL2926693 0.72 GABRA5 (0.56) GABRA5
SCHEMBL1776863 0.72 GABRA5 (0.48) GABRA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427455-A1 ISOXAZOLE-PYRAZOLE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2012-03-14 EP disclosed
WO-2010127975-A1 ISOXAZOLE-PYRAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2010-11-11 WO disclosed