SCHEMBL28628147

SCHEMBL28628147

O=C1CC2(CCOCC2)Oc2cc(Br)ccc21

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.48
CA2 P00918 2/20 0.48
CA7 P43166 2/20 0.48
CA9 Q16790 2/20 0.48
HTR2A P28223 1/20 0.48
HTR2C P28335 1/20 0.48
HDAC3 O15379 4/20 0.44
HDAC4 P56524 4/20 0.44
HDAC1 Q13547 4/20 0.44
HDAC7 Q8WUI4 4/20 0.44
HDAC2 Q92769 4/20 0.44
HDAC10 Q969S8 4/20 0.44
HDAC11 Q96DB2 4/20 0.44
HDAC8 Q9BY41 4/20 0.44
HDAC6 Q9UBN7 4/20 0.44
HDAC9 Q9UKV0 4/20 0.44
HDAC5 Q9UQL6 4/20 0.44
KDM4E B2RXH2 4/20 0.43
ATM Q13315 3/20 0.43
HTT P42858 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1819491 0.88 KDM4E (0.54) CA1CA2CA7CA9HDAC3
SCHEMBL7609327 0.88 KDM4E (0.56) CA1CA2CA7CA9HTR2A
SCHEMBL4781793 0.88 KDM4E (0.52) CA1CA2CA7CA9HTR2A
SCHEMBL28840807 0.87 KDM4E (0.57) CA1CA2CA7CA9HTR2A
SCHEMBL30953726 0.85 HTR2A (0.50) CA1CA2CA7CA9HTR2A
SCHEMBL13791454 0.84 HDAC3 (0.60) CA1CA2CA7CA9HTR2A
SCHEMBL7959375 0.83 KDM4E (0.56) CA1CA2CA7CA9HDAC3
SCHEMBL3953983 0.82 KDM4E (0.60) CA1CA2CA7CA9HTR2C
SCHEMBL4346066 0.82 HSD11B1 (0.45) HTR2AHDAC3HDAC4HDAC1HDAC7
SCHEMBL3594528 0.80 RAF1 (0.46) HDAC3HDAC4HDAC1HDAC7HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113429440-B Prodrug of spiro compound, preparation method and application thereof in medicine 江苏恒瑞医药股份有限公司 2023-05-12 CN disclosed
CN-113264945-B Spiro derivative, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2022-11-22 CN disclosed
CN-113429440-A Prodrug of spiro compound, preparation method and application thereof in medicine 江苏恒瑞医药股份有限公司 2021-09-24 CN disclosed
CN-113264945-A Spiro derivative, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2021-08-17 CN disclosed