SCHEMBL28628183

SCHEMBL28628183

O=C1CCc2cccc(CO)c2N1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.46
MAPK13 O15264 1/20 0.46
MAPK12 P53778 1/20 0.46
MAPK11 Q15759 1/20 0.46
MAPK14 Q16539 1/20 0.46
HTR2A P28223 1/20 0.45
SRD5A1 P18405 2/20 0.39
AHR P35869 1/20 0.39
CYP11B1 P15538 4/20 0.38
CYP11B2 P19099 4/20 0.38
CYP19A1 P11511 3/20 0.38
CRBN Q96SW2 3/20 0.37
DDB1 Q16531 1/20 0.37
KDM4E B2RXH2 1/20 0.36
MAPT P10636 1/20 0.36
BRD4 O60885 1/20 0.36
CA9 Q16790 1/20 0.34
KIF11 P52732 2/20 0.34
CYP1A2 P05177 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8284040 0.90 MAPT (0.49) NPC1MAPK13MAPK12MAPK11MAPK14
SCHEMBL17969062 0.84 NPC1 (0.47) NPC1MAPK13MAPK12MAPK11MAPK14
SCHEMBL8919270 0.84 NPC1 (0.47) NPC1MAPK13MAPK12MAPK11MAPK14
SCHEMBL11266794 0.83 NPC1 (0.46) NPC1MAPK13MAPK12MAPK11MAPK14
SCHEMBL10788798 0.82 NPC1 (0.42) NPC1MAPK13MAPK12MAPK11MAPK14
SCHEMBL10646325 0.80 PARP1 (0.43) NPC1MAPK13MAPK12MAPK11MAPK14
SCHEMBL20702475 0.78 NPC1 (0.41) NPC1MAPK13MAPK12MAPK11MAPK14
SCHEMBL2215753 0.77 SRD5A1 (0.37) NPC1MAPK13MAPK12MAPK11MAPK14
SCHEMBL29410901 0.77 NPC1 (0.50) NPC1MAPK13MAPK12MAPK11MAPK14
SCHEMBL2230502 0.77 NPC1 (0.50) NPC1MAPK13MAPK12MAPK11MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113429410-B Polyheterocyclic substituted pyrimidine or pyridylamine derivatives, compositions and medical uses thereof 上海海雁医药科技有限公司 2022-10-04 CN disclosed
CN-113429410-A Polyheterocyclic substituted pyrimidine or pyridylamine derivatives, compositions and medical uses thereof 上海海雁医药科技有限公司 2021-09-24 CN disclosed