SCHEMBL28628800

SCHEMBL28628800

CN(C)c1ccc(C#N)cc1C#Cc1ccccc1Br

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 2/20 0.36
ALDH1A1 P00352 4/20 0.36
KDM4E B2RXH2 1/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36
CXCR2 P25025 2/20 0.35
CXCR1 P25024 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.34
IMPDH2 P12268 1/20 0.32
IMPDH1 P20839 1/20 0.32
LRRK2 Q5S007 1/20 0.31
PGR P06401 2/20 0.31
KDM1A O60341 1/20 0.31
TSHR P16473 2/20 0.31
MEN1 O00255 1/20 0.31
LMNA P02545 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29893806 1.00 FFAR1 (0.36) FFAR1ALDH1A1KDM4EGAAMAPT
SCHEMBL8651599 0.77 ALDH1A1 (0.46) ALDH1A1KDM4EGAAMAPTIMPDH2
SCHEMBL1778656 0.76 MEN1 (0.42) ALDH1A1KDM4EGAAMAPTPGR
SCHEMBL29893809 0.75 PTPN1 (0.36) FFAR1GAAMAPTPTGDR2MEN1
SCHEMBL29894671 0.73 ALDH1A1 (0.46) ALDH1A1MAPTCXCR2CXCR1TSHR
SCHEMBL12408477 0.69 FFAR1 (0.59) FFAR1ALDH1A1KDM4EMAPTMEN1
SCHEMBL30468202 0.69 FFAR1 (0.47) FFAR1ALDH1A1KDM4EGAAMAPT
SCHEMBL2466535 0.69 FFAR1 (0.47) FFAR1ALDH1A1KDM4EGAAMAPT
SCHEMBL29894046 0.68 CA12 (0.33) ALDH1A1KDM4EGAAMAPTTSHR
SCHEMBL31235647 0.67 MEN1 (0.43) ALDH1A1CXCR2CXCR1IMPDH2IMPDH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113121542-B 5, 10-indolino [3,2-b ] indole derivative and synthetic method and application thereof 常州大学 2022-09-30 CN disclosed
CN-113372258-A Indeno [1,2-b ] indole derivative and preparation method and application thereof 常州大学 2021-09-10 CN disclosed
CN-113121542-A 5, 10-indolino [3,2-b ] indole derivative and synthesis method and application thereof 常州大学 2021-07-16 CN disclosed