SCHEMBL28629043

SCHEMBL28629043

CC(N)C(O)c1ncccn1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.46
LMNA P02545 4/20 0.46
HIF1A Q16665 3/20 0.46
ADRA2A P08913 1/20 0.46
ADRA2C P18825 1/20 0.46
ALDH1A1 P00352 1/20 0.45
APLNR P35414 1/20 0.40
ADRB1 P08588 1/20 0.39
MIF P14174 1/20 0.39
HTR2A P28223 1/20 0.39
ADRA1A P35348 1/20 0.39
HTR2B P41595 1/20 0.39
RECQL P46063 4/20 0.36
TDP1 Q9NUW8 4/20 0.36
MAPT P10636 3/20 0.36
ALOX15 P16050 1/20 0.36
TSHR P16473 1/20 0.36
NFKB1 P19838 1/20 0.36
THPO P40225 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16492788 1.00 KDM4E (0.46) KDM4ELMNAHIF1AADRA2AADRA2C
SCHEMBL28266841 0.80 APLNR (0.43) KDM4ELMNAHIF1AADRA2AADRA2C
SCHEMBL1856675 0.75 HSP90AA1 (0.35) KDM4ELMNAHIF1AADRA2AADRA2C
SCHEMBL5227874 0.74 KDM4E (0.50) KDM4ELMNAHIF1AADRA2AADRA2C
SCHEMBL4969094 0.74 KDM4E (0.50) KDM4ELMNAHIF1AADRA2AADRA2C
SCHEMBL310530 0.74
SCHEMBL20567997 0.74
SCHEMBL21031336 0.74
SCHEMBL26917162 0.74
SCHEMBL7352602 0.74

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106661084-B Macrocyclic broad spectrum antibiotics 阿奇克斯制药公司 2021-08-31 CN disclosed