Quinazoline

Quinazoline

SCHEMBL28634018

O=Cc1ccccc1.c1ccc2ncncc2c1

nearest known ligand 0.69

Full drug profile on Sugi Atlas →

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
EGFR P00533 9/20 0.69
ALDH1A1 P00352 1/20 0.48
CYP2A6 P11509 1/20 0.48
PIK3CD O00329 1/20 0.47
PIK3CA P42336 1/20 0.47
PDGFRB P09619 1/20 0.45
PDGFRA P16234 1/20 0.45
RAB9A P51151 1/20 0.40
FGFR1 P11362 1/20 0.38
MGAM O43451 1/20 0.38
IMPDH2 P12268 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Quinoline SCHEMBL28247366 0.92 EGFR (0.59) EGFRALDH1A1CYP2A6PIK3CDPIK3CA
SCHEMBL3196932 0.85 EGFR (0.95) EGFRALDH1A1PIK3CDPIK3CAPDGFRB
Quinazoline SCHEMBL29902476 0.84 EGFR (0.77) EGFRALDH1A1PIK3CDPIK3CAPDGFRB
Quinazoline SCHEMBL1337802 0.84 EGFR (0.77) EGFRALDH1A1PIK3CDPIK3CAPDGFRB
Quinazoline SCHEMBL29490398 0.83 EGFR (1.00) EGFRALDH1A1CYP2A6PIK3CDPIK3CA
Quinazoline SCHEMBL29356169 0.83 EGFR (1.00) EGFRALDH1A1CYP2A6PIK3CDPIK3CA
Quinazoline SCHEMBL22833783 0.83 EGFR (1.00) EGFRALDH1A1CYP2A6PIK3CDPIK3CA
Quinazoline SCHEMBL5920 0.83 EGFR (1.00) EGFRALDH1A1CYP2A6PIK3CDPIK3CA
Quinazoline SCHEMBL27762358 0.83 EGFR (0.69) EGFRALDH1A1PIK3CDPIK3CAPDGFRB
Quinazoline SCHEMBL27786386 0.81 EGFR (0.87) EGFRALDH1A1CYP2A6PIK3CDPIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108699040-B Modulators of CFTR and methods of use thereof 加利福尼亚大学董事会 2021-08-10 CN disclosed