SCHEMBL28635642

SCHEMBL28635642

COC(=O)c1nc(-c2cccc(Br)c2C)oc1SC

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.41
HSD17B10 Q99714 5/20 0.41
PPARG P37231 2/20 0.41
NCOA2 Q15596 1/20 0.41
ALDH1A1 P00352 6/20 0.38
HPGD P15428 4/20 0.38
PKM P14618 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
L3MBTL1 Q9Y468 2/20 0.36
TOP2A P11388 2/20 0.36
IKBKB O14920 2/20 0.34
VDR P11473 2/20 0.34
MAPT P10636 6/20 0.34
TP53 P04637 4/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
NPC1 O15118 1/20 0.34
NFKB1 P19838 1/20 0.34
RAB9A P51151 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30703771 1.00 KDM4E (0.41) KDM4EHSD17B10PPARGNCOA2ALDH1A1
SCHEMBL30703864 0.86 KDM4E (0.44) KDM4EHSD17B10PPARGNCOA2ALDH1A1
SCHEMBL28652254 0.86 KDM4E (0.44) KDM4EHSD17B10PPARGNCOA2ALDH1A1
SCHEMBL30703825 0.78 ALDH1A1 (0.36) KDM4EHSD17B10PPARGNCOA2ALDH1A1
SCHEMBL22308216 0.78 ALDH1A1 (0.53) KDM4EHSD17B10PPARGALDH1A1HPGD
SCHEMBL28647095 0.78 ALDH1A1 (0.36) KDM4EHSD17B10PPARGNCOA2ALDH1A1
SCHEMBL31521809 0.78 ALDH1A1 (0.53) KDM4EHSD17B10PPARGALDH1A1HPGD
SCHEMBL21842992 0.75 TP53 (0.44) KDM4EHSD17B10ALDH1A1HPGDNPSR1
SCHEMBL23198773 0.72 MAPT (0.54) KDM4EHSD17B10ALDH1A1HPGDL3MBTL1
SCHEMBL20295983 0.70 TOP2A (0.47) KDM4EHSD17B10ALDH1A1HPGDNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113348170-B Biphenyl derivative inhibitor, preparation method and application thereof 上海翰森生物医药科技有限公司 2023-12-22 CN disclosed
CN-113348170-A Biphenyl derivative inhibitor, preparation method and application thereof 上海翰森生物医药科技有限公司 2021-09-03 CN disclosed