SCHEMBL28635699

SCHEMBL28635699

COC(=O)c1ccc(CN(C(=O)N2CCSCC2)c2cccc(-c3ccc4cnn(C)c4c3)c2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FASN P49327 1/20 0.40
TNKS O95271 2/20 0.40
TNKS2 Q9H2K2 2/20 0.40
HDAC1 Q13547 2/20 0.38
HDAC6 Q9UBN7 2/20 0.38
HDAC8 Q9BY41 1/20 0.38
PIK3CA P42336 1/20 0.37
QPCT Q16769 1/20 0.36
PDE1C Q14123 1/20 0.35
AGTR1 P30556 1/20 0.35
NR1H4 Q96RI1 2/20 0.35
AR P10275 1/20 0.34
SCD5 Q86SK9 1/20 0.34
CYP19A1 P11511 1/20 0.34
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34
DRD2 P14416 1/20 0.34
TBXA2R P21731 1/20 0.34
MGLL Q99685 1/20 0.34
MKNK1 Q9BUB5 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28628419 0.93 TNKS (0.46) FASNTNKSTNKS2PIK3CAQPCT
SCHEMBL16211835 0.90 HDAC1 (0.48) FASNTNKSTNKS2HDAC1HDAC6
SCHEMBL22218170 0.90 TNKS (0.40) FASNTNKSTNKS2HDAC1HDAC6
SCHEMBL22218172 0.90 TNKS (0.40) FASNTNKSTNKS2HDAC1HDAC6
SCHEMBL16211361 0.86 TNKS (0.42) FASNTNKSTNKS2HDAC1HDAC6
SCHEMBL16211520 0.86 TNKS (0.42) FASNTNKSTNKS2HDAC1HDAC6
SCHEMBL28641692 0.85 CETP (0.43) HDAC1HDAC6HDAC8NR1H4AR
SCHEMBL16213193 0.85 HDAC1 (0.48) TNKSTNKS2HDAC1HDAC6HDAC8
SCHEMBL16211339 0.83 TNKS (0.46) FASNTNKSTNKS2HDAC1HDAC6
SCHEMBL22218669 0.82 TNKS (0.45) FASNTNKSTNKS2PIK3CAQPCT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108137518-B 1,3, 4-oxadiazole derivative compounds as histone deacetylase 6 inhibitors and pharmaceutical compositions comprising the same 株式会社钟根堂 2021-08-31 CN disclosed