SCHEMBL28628419

SCHEMBL28628419

COC(=O)c1ccc(CN(C(=O)N2CCSCC2)c2ccc(-c3ccc4cnn(C)c4c3)cc2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNKS O95271 2/20 0.46
TNKS2 Q9H2K2 2/20 0.46
FASN P49327 1/20 0.44
PIK3CA P42336 1/20 0.39
NR1H4 Q96RI1 2/20 0.37
QPCT Q16769 1/20 0.37
PDE1C Q14123 1/20 0.36
CHKA P35790 1/20 0.36
AR P10275 1/20 0.36
CTSC P53634 1/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
MKNK1 Q9BUB5 1/20 0.35
MKNK2 Q9HBH9 1/20 0.35
ERCC1 P07992 1/20 0.35
ERCC4 Q92889 1/20 0.35
AGTR1 P30556 1/20 0.35
MLYCD O95822 1/20 0.35
PTGER3 P43115 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28635699 0.93 FASN (0.40) TNKSTNKS2FASNPIK3CANR1H4
SCHEMBL16211339 0.90 TNKS (0.46) TNKSTNKS2FASNPIK3CANR1H4
SCHEMBL22218671 0.89 TNKS (0.45) TNKSTNKS2FASNPIK3CANR1H4
SCHEMBL22218669 0.89 TNKS (0.45) TNKSTNKS2FASNPIK3CANR1H4
SCHEMBL20236846 0.86 FASN (0.42) TNKSTNKS2FASNPIK3CAQPCT
SCHEMBL28637466 0.83 PTGES (0.43) NR1H4CHKAARRAB9A
SCHEMBL16211835 0.83 HDAC1 (0.48) TNKSTNKS2FASNPIK3CARAB9A
SCHEMBL22218172 0.82 TNKS (0.40) TNKSTNKS2FASNPIK3CANR1H4
SCHEMBL22218170 0.82 TNKS (0.40) TNKSTNKS2FASNPIK3CANR1H4
SCHEMBL28632493 0.81 TNKS (0.43) TNKSTNKS2FASNQPCTPDE1C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108137518-B 1,3, 4-oxadiazole derivative compounds as histone deacetylase 6 inhibitors and pharmaceutical compositions comprising the same 株式会社钟根堂 2021-08-31 CN disclosed