SCHEMBL28636724

SCHEMBL28636724

Cc1cc(Nc2ccnc([S+]([O-])Cc3ccc(C(=O)O)cc3)n2)n[nH]1

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ITK Q08881 1/20 0.48
IGF1R P08069 3/20 0.43
FGFR1 P11362 3/20 0.43
KDR P35968 3/20 0.43
AURKA O14965 6/20 0.43
AURKB Q96GD4 2/20 0.43
EGFR P00533 2/20 0.42
CCNA2 P20248 2/20 0.40
CDK2 P24941 2/20 0.40
CCNA1 P78396 2/20 0.40
RET P07949 4/20 0.38
PIK3C3 Q8NEB9 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28639456 0.82 HDAC1 (0.53) RET
SCHEMBL30363242 0.82 HDAC1 (0.53) RET
SCHEMBL23963005 0.79 ITK (0.53) ITKIGF1RFGFR1KDRAURKA
SCHEMBL23929024 0.78 AURKA (0.53) ITKIGF1RFGFR1KDRAURKA
SCHEMBL23962996 0.68 AURKA (0.52) ITKKDRAURKAAURKB
SCHEMBL18154707 0.67 ITK (0.65) ITKIGF1RFGFR1KDRAURKA
SCHEMBL30230471 0.67 ITK (0.65) ITKIGF1RFGFR1KDRAURKA
SCHEMBL23963003 0.67 ITK (0.44) ITKIGF1RFGFR1KDRAURKA
SCHEMBL18297012 0.65 ITK (0.50) ITKIGF1RFGFR1KDRAURKA
SCHEMBL5766890 0.65 IGF1R (0.50) ITKIGF1RFGFR1KDRAURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113549057-B Snail inhibitor and derivative thereof, preparation method, pharmaceutical composition and application 中国药科大学 2023-01-31 CN disclosed
CN-113549057-A Snail inhibitor and derivative thereof, preparation method, pharmaceutical composition and application 中国药科大学 2021-10-26 CN disclosed