SCHEMBL23963003

SCHEMBL23963003

CC/C=C\CC(C)[S@@+]([O-])c1nccc(Nc2cc(C)[nH]n2)n1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ITK Q08881 1/20 0.44
IGF1R P08069 6/20 0.41
KDR P35968 5/20 0.41
FGFR1 P11362 4/20 0.41
AURKA O14965 5/20 0.37
AURKB Q96GD4 4/20 0.37
EGFR P00533 3/20 0.37
JAK2 O60674 2/20 0.34
JAK3 P52333 2/20 0.34
INSR P06213 1/20 0.34
SRC P12931 1/20 0.34
FLT4 P35916 1/20 0.34
PIK3C3 Q8NEB9 1/20 0.34
DHODH Q02127 1/20 0.33
CYP2D6 P10635 1/20 0.33
PKN1 Q16512 1/20 0.33
NTRK1 P04629 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23963005 0.78 ITK (0.53) ITKIGF1RKDRFGFR1AURKA
SCHEMBL18154707 0.68 ITK (0.65) ITKIGF1RKDRFGFR1AURKA
SCHEMBL30230471 0.68 ITK (0.65) ITKIGF1RKDRFGFR1AURKA
SCHEMBL28636724 0.67 ITK (0.48) ITKIGF1RKDRFGFR1AURKA
SCHEMBL18154760 0.67 ITK (0.56) ITKIGF1RKDRFGFR1AURKA
SCHEMBL30353181 0.66 ITK (0.55) ITKIGF1RKDRFGFR1AURKA
SCHEMBL2120764 0.66 ITK (0.62) ITKIGF1RKDRFGFR1AURKA
SCHEMBL29537888 0.66 ITK (0.62) ITKIGF1RKDRFGFR1AURKA
SCHEMBL13675364 0.64 ITK (0.56) ITKIGF1RKDRFGFR1AURKA
SCHEMBL18154778 0.64 ITK (0.59) ITKIGF1RKDRFGFR1AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021213111-A1 SNAIL INHIBITOR, DERIVATIVE THEREOF, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND USE THEREOF 中国药科大学 (CN) 2021-10-28 WO disclosed