SCHEMBL28637601

SCHEMBL28637601

CC(C)n1cc(-c2sc(N)nc2-c2c(F)cccc2F)ccc1=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 5/20 0.46
ADORA1 P30542 4/20 0.46
ADORA2B P29275 3/20 0.42
ADORA3 P0DMS8 1/20 0.42
BMPR1B O00238 2/20 0.38
BMPR1A P36894 2/20 0.38
TGFBR1 P36897 2/20 0.38
ACVRL1 P37023 2/20 0.38
ACVR1 Q04771 2/20 0.38
MAPT P10636 3/20 0.38
KDM4E B2RXH2 2/20 0.38
LMNA P02545 2/20 0.38
MAPK1 P28482 2/20 0.38
XBP1 P17861 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
ATR Q13535 7/20 0.37
ALDH1A1 P00352 3/20 0.37
CYP1A2 P05177 2/20 0.37
CYP2D6 P10635 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28637600 0.88 ADORA2A (0.44) ADORA2AADORA1ADORA2BADORA3BMPR1B
SCHEMBL28637603 0.87 ADORA2A (0.46) ADORA2AADORA1ADORA2BADORA3BMPR1B
SCHEMBL28646803 0.84 ADORA2A (0.61) ADORA2AADORA1ADORA2BADORA3BMPR1B
SCHEMBL28658385 0.84 ADORA2A (0.47) ADORA2AADORA1BMPR1BBMPR1ATGFBR1
SCHEMBL28647185 0.84 ADORA2A (0.46) ADORA2AADORA1ADORA2BADORA3BMPR1B
SCHEMBL28645614 0.83 ADORA2A (0.51) ADORA2AADORA1ADORA2BADORA3BMPR1B
SCHEMBL28637791 0.83 ALDH1A1 (0.57) ADORA2AADORA1MAPTKDM4ELMNA
SCHEMBL28645393 0.81 ADORA2A (0.49) ADORA2AADORA1ADORA2BADORA3BMPR1B
SCHEMBL28926809 0.81 ADORA2A (0.49) ADORA2AADORA1ADORA2BADORA3BMPR1B
SCHEMBL28642914 0.80 MAPT (0.47) ADORA2AADORA1BMPR1BBMPR1ATGFBR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109293652-B Substituted thiazole derivative and application thereof 四川科伦博泰生物医药股份有限公司 2021-10-22 CN disclosed