SCHEMBL28638045

SCHEMBL28638045

O=Cc1cn2c(n1)CN(Cc1ccc(C(=O)O)cc1)CC2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.43
THRB P10828 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
LMNA P02545 1/20 0.43
HDAC6 Q9UBN7 2/20 0.42
KDM1A O60341 1/20 0.42
HDAC4 P56524 2/20 0.40
HDAC1 Q13547 2/20 0.40
KCNH2 Q12809 1/20 0.40
HSD17B10 Q99714 1/20 0.40
COMT P21964 1/20 0.39
LTA4H P09960 4/20 0.38
GRM2 Q14416 1/20 0.37
NPC1 O15118 1/20 0.37
ALDH1A1 P00352 2/20 0.36
HDAC3 O15379 1/20 0.36
HDAC7 Q8WUI4 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC10 Q969S8 1/20 0.36
HDAC11 Q96DB2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2923547 0.87 COMT (0.46) GAASMN1; SMN2LMNAHSD17B10COMT
SCHEMBL19586255 0.86 GAA (0.47) GAASMN1; SMN2HDAC6KDM1AALDH1A1
SCHEMBL28642452 0.74 KDM1A (0.49) GAASMN1; SMN2LMNAHDAC6KDM1A
SCHEMBL6382726 0.74 HRH4 (0.31)
SCHEMBL10074441 0.72 HDAC1 (0.62) GAATHRBSMN1; SMN2LMNAHDAC6
SCHEMBL27519383 0.71 HDAC4 (0.71) SMN1; SMN2LMNAHDAC4HDAC1KCNH2
SCHEMBL2926205 0.70 COMT (0.37) COMT
SCHEMBL29275413 0.69 HDAC4 (0.55) GAATHRBSMN1; SMN2LMNAHDAC6
SCHEMBL19609092 0.69 KDM1A (0.49) GAASMN1; SMN2LMNAHDAC6KDM1A
SCHEMBL14217257 0.69 HDAC1 (0.54) GAATHRBSMN1; SMN2LMNAHDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109153636-B Cyclopropyl-amide compounds as dual LSD1/HDAC inhibitors 朱比连特埃皮科尔有限责任公司 2021-10-22 CN disclosed