SCHEMBL28638558

SCHEMBL28638558

CCOC(=O)c1cc2c(cc1OCC)C(=O)N(CC1CCN(C(C)=O)CC1)C2

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 1/20 0.41
UGCG Q16739 1/20 0.41
REV1 Q9UBZ9 1/20 0.39
AKR1C3 P42330 1/20 0.38
AKR1C2 P52895 1/20 0.38
MAPT P10636 2/20 0.38
PRMT5 O14744 2/20 0.36
WDR77 Q9BQA1 1/20 0.36
LMNA P02545 1/20 0.36
F10 P00742 2/20 0.36
TP53 P04637 1/20 0.35
GLA P06280 1/20 0.35
KCNK3 O14649 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
PARP1 P09874 1/20 0.35
PARP2 Q9UGN5 1/20 0.35
HSP90AA1 P07900 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30604562 1.00 NR1I2 (0.41) NR1I2UGCGREV1AKR1C3AKR1C2
SCHEMBL30604573 0.92 NR1I2 (0.42) NR1I2UGCGAKR1C3AKR1C2LMNA
SCHEMBL28638409 0.92 NR1I2 (0.42) NR1I2UGCGAKR1C3AKR1C2LMNA
SCHEMBL28639020 0.89 HPGD (0.45) NR1I2UGCGMAPTLMNATP53
SCHEMBL30604610 0.89 HPGD (0.45) NR1I2UGCGMAPTLMNATP53
SCHEMBL30604560 0.87 IRAK4 (0.43) NR1I2UGCGAKR1C3AKR1C2LMNA
SCHEMBL28638399 0.87 IRAK4 (0.43) NR1I2UGCGAKR1C3AKR1C2LMNA
SCHEMBL28645369 0.87 PARP1 (0.44) NR1I2UGCGAKR1C3AKR1C2LMNA
SCHEMBL28645772 0.78 PARP1 (0.40) AKR1C3AKR1C2MAPTTP53KCNK3
SCHEMBL28926168 0.78 MEN1 (0.39) AKR1C3AKR1C2MAPTLMNATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113493438-B Tetrahydroisoquinoline compounds 南京再明医药有限公司 2023-10-20 CN disclosed
CN-113493438-A Tetrahydroisoquinoline compounds 江苏先声药业有限公司 2021-10-12 CN disclosed