SCHEMBL28645772

SCHEMBL28645772

CCOC(=O)c1cc2c(cc1OCC)C(=O)N(CC(C)C)C2

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
HSP90AA1 P07900 1/20 0.39
AKR1C3 P42330 1/20 0.38
AKR1C2 P52895 1/20 0.38
ALDH1A1 P00352 2/20 0.38
KCNK3 O14649 1/20 0.37
KDM4E B2RXH2 2/20 0.36
PKM P14618 1/20 0.36
GABRA1 P14867 2/20 0.36
MAPT P10636 2/20 0.36
TP53 P04637 1/20 0.36
IRAK4 Q9NWZ3 1/20 0.35
NPC1 O15118 1/20 0.35
POLB P06746 1/20 0.35
IDH1 O75874 1/20 0.35
GABRG2 P18507 1/20 0.35
GABRB3 P28472 1/20 0.35
GABRA5 P31644 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28645763 0.88 KMT2A (0.41) PARP1MEN1KMT2ANPC1POLB
SCHEMBL28926168 0.84 MEN1 (0.39) MEN1KMT2AHSP90AA1AKR1C3AKR1C2
SCHEMBL28639031 0.81 KMT2A (0.57) PARP1MEN1KMT2AHSP90AA1ALDH1A1
SCHEMBL30604573 0.80 NR1I2 (0.42) PARP1MEN1KMT2AAKR1C3AKR1C2
SCHEMBL28656587 0.80 TSHR (0.51) PARP1MEN1KMT2AHSP90AA1MAPT
SCHEMBL28638409 0.80 NR1I2 (0.42) PARP1MEN1KMT2AAKR1C3AKR1C2
SCHEMBL28645766 0.80 MEN1 (0.53) MEN1KMT2AALDH1A1KDM4EPKM
SCHEMBL30604599 0.80 MEN1 (0.53) MEN1KMT2AALDH1A1KDM4EPKM
SCHEMBL28925117 0.80 MEN1 (0.50) MEN1KMT2AALDH1A1GABRA1MAPT
SCHEMBL28638399 0.79 IRAK4 (0.43) MEN1KMT2AAKR1C3AKR1C2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113493438-B Tetrahydroisoquinoline compounds 南京再明医药有限公司 2023-10-20 CN disclosed
CN-113493438-A Tetrahydroisoquinoline compounds 江苏先声药业有限公司 2021-10-12 CN disclosed