SCHEMBL28644181

SCHEMBL28644181

N#Cc1cccc(-c2nccc3c2[nH]c2ccc(F)cc23)c1

nearest known ligand 0.74

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TDO2 P48775 9/20 0.74
BCHE P06276 3/20 0.52
IDO1 P14902 5/20 0.49
HTR2B P41595 2/20 0.47
HTR5A P47898 2/20 0.47
AR P10275 1/20 0.44
CLK4 Q9HAZ1 2/20 0.42
CLK1 P49759 1/20 0.42
CLK2 P49760 1/20 0.42
DYRK1A Q13627 1/20 0.42
DYRK1B Q9Y463 1/20 0.42
PARP1 P09874 1/20 0.41
PARP3 Q9Y6F1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30923483 1.00 TDO2 (0.74) TDO2BCHEIDO1HTR2BHTR5A
SCHEMBL28651658 0.91 TDO2 (0.74) TDO2BCHEIDO1HTR2BHTR5A
SCHEMBL30923488 0.91 TDO2 (0.74) TDO2BCHEIDO1HTR2BHTR5A
SCHEMBL30923490 0.82 TDO2 (0.73) TDO2BCHEIDO1HTR2BHTR5A
SCHEMBL28639491 0.82 TDO2 (0.73) TDO2BCHEIDO1HTR2BHTR5A
SCHEMBL28644260 0.82 TDO2 (0.73) TDO2BCHEIDO1HTR2BHTR5A
SCHEMBL30923477 0.82 TDO2 (0.73) TDO2BCHEIDO1HTR2BHTR5A
SCHEMBL30923486 0.77 IDO1 (0.76) TDO2BCHEIDO1HTR2BHTR5A
SCHEMBL28657328 0.77 IDO1 (0.76) TDO2BCHEIDO1HTR2BHTR5A
SCHEMBL29130513 0.76 TDO2 (1.00) TDO2BCHEIDO1HTR2BHTR5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113307806-B Beta-carboline selective monoamine oxidase B inhibitor and pharmaceutical application thereof 南京医科大学 2024-05-14 CN disclosed
CN-113307806-A Beta-carboline selective monoamine oxidase B inhibitor and pharmaceutical application thereof 陈冬寅 2021-08-27 CN disclosed