SCHEMBL28646753

SCHEMBL28646753

Fc1ccc(-c2[c]nccn2)c(Cl)c1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 1/20 0.43
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
HSD11B1 P28845 2/20 0.38
MAPK14 Q16539 6/20 0.37
GRM2 Q14416 2/20 0.35
GCGR P47871 1/20 0.35
CYP17A1 P05093 1/20 0.33
CLK1 P49759 1/20 0.33
ROS1 P08922 1/20 0.32
ABL1 P00519 1/20 0.32
KDM4E B2RXH2 1/20 0.32
TP53 P04637 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
CNR1 P21554 1/20 0.31
CNR2 P34972 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28635233 0.83 EGLN2 (0.41) NPC1RAB9AHSD11B1KDM4ETP53
SCHEMBL28635232 0.80 HSP90AB1 (0.35) NISCHMAPK14
SCHEMBL22261806 0.71 CCNB2 (0.37) NPC1RAB9AMAPK14GCGR
SCHEMBL28632034 0.70 GRM2 (0.35) NISCHGRM2
SCHEMBL7500881 0.69 CYP17A1 (0.42) NISCHCYP17A1KDM4E
SCHEMBL1688524 0.69 NISCH (0.49) NISCHNPC1RAB9AHSD11B1MAPK14
SCHEMBL22261800 0.68 NOTUM (0.38) NISCHNPC1KDM4E
SCHEMBL450465 0.66
SCHEMBL3383277 0.66 MAPK14 (0.56) NISCHMAPK14GCGR
SCHEMBL22310234 0.66 NISCH (0.42) NISCHNPC1RAB9AHSD11B1MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108026050-B Novel compounds as ROR gamma modulators 格兰马克药品股份有限公司 2021-04-30 CN disclosed