SCHEMBL28635233

SCHEMBL28635233

Clc1ccc(-c2[c]nccn2)c(Cl)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGLN2 Q96KS0 2/20 0.41
AHR P35869 1/20 0.40
HSD11B1 P28845 2/20 0.40
GRM5 P41594 1/20 0.39
MAPT P10636 3/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
PIK3CA P42336 1/20 0.38
PIK3CB P42338 1/20 0.38
PIK3CG P48736 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
ALDH1A1 P00352 3/20 0.37
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
PKM P14618 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
HSP90AA1 P07900 1/20 0.37
HSP90AB1 P08238 1/20 0.37
KDM4E B2RXH2 1/20 0.37
MGAM O43451 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28646753 0.83 NISCH (0.43) HSD11B1SMN1; SMN2NPC1RAB9AKDM4E
SCHEMBL1275106 0.74 MAPT (0.42) EGLN2AHRHSD11B1GRM5MAPT
SCHEMBL22261807 0.73 CCNB2 (0.37) MAPTMEN1KMT2ANPC1RAB9A
SCHEMBL29624840 0.68 AHR (0.64) AHRHSD11B1MAPTALDH1A1RAB9A
SCHEMBL464507 0.68 AHR (0.64) AHRHSD11B1MAPTALDH1A1RAB9A
SCHEMBL28630972 0.68 LMNA (0.36) MAPTMEN1KMT2ASMN1; SMN2ALDH1A1
SCHEMBL3453300 0.67 GRM5 (0.51) EGLN2AHRHSD11B1GRM5MAPT
SCHEMBL3631532 0.67 RAB9A (0.50) EGLN2AHRHSD11B1MAPTMEN1
SCHEMBL28635232 0.66 HSP90AB1 (0.35) GRM5HSP90AB1
SCHEMBL28632034 0.66 GRM2 (0.35) GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108026050-B Novel compounds as ROR gamma modulators 格兰马克药品股份有限公司 2021-04-30 CN disclosed