SCHEMBL28648124

SCHEMBL28648124

COc1ccc(C(=O)Cl)cc1-n1cnc(C2CC2)c1

nearest known ligand 0.42

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MAP3K5 Q99683 16/20 0.42
ABL1 P00519 2/20 0.40
LMNA P02545 1/20 0.36
HPGD P15428 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28657015 0.89 TSHR (0.45) MAP3K5ABL1LMNAHPGD
SCHEMBL28643381 0.88 MAPK1 (0.43) MAP3K5ABL1LMNA
SCHEMBL28649133 0.88 MAP3K5 (0.44) MAP3K5ABL1HPGD
SCHEMBL28643374 0.84 MAP3K5 (0.52) MAP3K5
SCHEMBL20750911 0.84 MAP3K5 (0.41) MAP3K5ABL1
SCHEMBL28660361 0.81 MAP3K5 (0.43) MAP3K5
SCHEMBL28658684 0.81 MAP3K5 (0.40) MAP3K5ABL1
SCHEMBL23865349 0.80 MAP3K5 (0.48) MAP3K5
SCHEMBL28643811 0.79 MAP3K5 (0.43) MAP3K5ABL1
SCHEMBL28658681 0.78 TLR2 (0.44) MAP3K5ABL1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109400625-B Fused bicyclic compound and application thereof in medicine 广东东阳光药业有限公司 2021-11-12 CN disclosed