SCHEMBL28657015

SCHEMBL28657015

COc1ccc(C(=O)O)cc1-n1cnc(C2CC2)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.45
HPGD P15428 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA4 P22748 1/20 0.44
CA6 P23280 1/20 0.44
CA7 P43166 1/20 0.44
TPMT P51580 1/20 0.44
CA9 Q16790 1/20 0.44
CA14 Q9ULX7 1/20 0.44
MAP3K5 Q99683 6/20 0.43
HTT P42858 2/20 0.42
LMNA P02545 1/20 0.42
MAPK1 P28482 1/20 0.42
RAB9A P51151 1/20 0.42
PDE4D Q08499 2/20 0.41
KDM4E B2RXH2 1/20 0.40
HSP90AA1 P07900 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28643381 0.89 MAPK1 (0.43) MAP3K5LMNAMAPK1PDE4DHSP90AA1
SCHEMBL28649133 0.89 MAP3K5 (0.44) HPGDNPSR1MAP3K5RAB9APDE4D
SCHEMBL28648124 0.89 MAP3K5 (0.42) HPGDMAP3K5LMNAABL1
SCHEMBL28649418 0.84 MAP3K5 (0.53) MAP3K5
SCHEMBL28656973 0.83 TSHR (0.41) TSHRMAP3K5HSD17B10ABL1KDM4C
SCHEMBL28658716 0.81 MAP3K5 (0.41) MAP3K5
SCHEMBL29949144 0.81 MAP3K5 (0.41) MAP3K5
SCHEMBL28648138 0.81 MAP3K5 (0.41) MAP3K5HSD17B10ABL1KDM4C
Hydrochloric Acid SCHEMBL28656984 0.80 MAP3K5 (0.41) MAP3K5
SCHEMBL22474009 0.79 MAP3K5 (0.49) MAP3K5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109400625-B Fused bicyclic compound and application thereof in medicine 广东东阳光药业有限公司 2021-11-12 CN disclosed