SCHEMBL28649192

SCHEMBL28649192

O=C(Nc1ccccc1)N1CCSCC1F

nearest known ligand 0.57

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.48
RAB9A P51151 3/20 0.48
SMN1; SMN2 Q16637 3/20 0.48
POLB P06746 2/20 0.45
KDM4E B2RXH2 3/20 0.44
TP53 P04637 2/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
MAPT P10636 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
LMNA P02545 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28653181 0.83 NPC1 (0.48) NPC1RAB9ASMN1; SMN2POLBKDM4E
SCHEMBL28637114 0.82 NPSR1 (0.46) NPC1RAB9ASMN1; SMN2POLBKDM4E
SCHEMBL28651312 0.80 POLB (0.45) NPC1RAB9ASMN1; SMN2POLBKDM4E
SCHEMBL31026228 0.74 RIPK1 (0.61) NPC1RAB9ASMN1; SMN2POLBKDM4E
SCHEMBL20236266 0.73 CYP2C9 (0.65) NPC1RAB9ASMN1; SMN2POLBKDM4E
SCHEMBL9984763 0.71 DPP4 (0.33)
SCHEMBL11145541 0.68 NPC1 (0.54) NPC1RAB9ASMN1; SMN2POLBKDM4E
SCHEMBL29155610 0.68 HPGD (0.60) NPC1RAB9ASMN1; SMN2POLBKDM4E
SCHEMBL2897923 0.67 KDM4E (0.77) SMN1; SMN2POLBKDM4ECYP2C9CYP2C19
SCHEMBL10729724 0.67 KDM4E (0.77) SMN1; SMN2POLBKDM4ECYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113651799-B Six-membered non-aromatic ring-containing diaryl pyrimidine HIV-1 reverse transcriptase inhibitor and preparation method and application thereof 山东大学 2022-06-17 CN disclosed
CN-113651799-A Six-membered non-aromatic ring-containing diaryl pyrimidine HIV-1 reverse transcriptase inhibitor and preparation method and application thereof 山东大学 2021-11-16 CN disclosed