SCHEMBL2865002

SCHEMBL2865002

Cc1nnc(-c2csc(-c3c(C)nc(-c4ncccc4O)n(CCc4ccccc4)c3=O)c2)o1

nearest known ligand 0.43

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
CASR P41180 19/20 0.43
NR1I2 O75469 4/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2858671 0.88 BRD4 (0.43) CASRNR1I2
SCHEMBL3418288 0.82 CASR (0.66) CASRNR1I2
SCHEMBL2839040 0.78 CASR (0.63) CASRNR1I2
SCHEMBL3418275 0.78 NR1I2 (0.51) CASRNR1I2
SCHEMBL3417598 0.75 CASR (0.60) CASRNR1I2
SCHEMBL2840722 0.74 CASR (0.73) CASRNR1I2
SCHEMBL3418557 0.74 NR1I2 (0.66) CASRNR1I2
Hydrochloric Acid SCHEMBL2835851 0.74 CASR (0.72) CASRNR1I2
SCHEMBL3421350 0.73 NR1I2 (0.63) CASRNR1I2
SCHEMBL2835550 0.73 CASR (0.61) CASRNR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010039913-A1 CALCILYTIC COMPOUNDS GLAXOSMITHKLINE LLC (US) 2010-04-08 WO claimed
WO-2010039913-A1 CALCILYTIC COMPOUNDS GLAXOSMITHKLINE LLC (US) 2010-04-08 WO disclosed
WO-2010039913-A1 CALCILYTIC COMPOUNDS GLAXOSMITHKLINE LLC (US) 2010-04-08 WO disclosed