SCHEMBL2858671

SCHEMBL2858671

Cc1nnc(-c2csc(-c3c(C)nc(-c4ncccc4OCc4ccccc4)n(CCc4ccccc4)c3=O)c2)o1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.43
CASR P41180 8/20 0.39
NR1I2 O75469 4/20 0.39
ALDH1A1 P00352 3/20 0.36
LMNA P02545 2/20 0.36
TSHR P16473 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
HIF1A Q16665 1/20 0.36
PTGER1 P34995 5/20 0.35
PTGER4 P35408 5/20 0.35
PTGER3 P43115 5/20 0.35
PTGER2 P43116 5/20 0.35
KDM4E B2RXH2 1/20 0.35
USP2 O75604 1/20 0.35
HSD17B10 Q99714 1/20 0.35
GCK P35557 1/20 0.34
SGMS2 Q8NHU3 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2865002 0.88 CASR (0.43) CASRNR1I2
SCHEMBL3418275 0.82 NR1I2 (0.51) BRD4CASRNR1I2ALDH1A1LMNA
SCHEMBL2838847 0.80 CASR (0.55) CASRNR1I2ALDH1A1LMNATSHR
SCHEMBL2837296 0.78 CASR (0.49) CASRNR1I2ALDH1A1LMNATSHR
SCHEMBL3418288 0.77 CASR (0.66) CASRNR1I2
SCHEMBL2835830 0.76 CASR (0.66) BRD4CASRNR1I2ALDH1A1LMNA
SCHEMBL4135738 0.75 CASR (0.49) BRD4CASRNR1I2ALDH1A1LMNA
SCHEMBL2839722 0.75 TSHR (0.46) CASRNR1I2ALDH1A1LMNATSHR
SCHEMBL3419476 0.74 NR1I2 (0.54) CASRNR1I2ALDH1A1LMNATSHR
SCHEMBL3421089 0.74 NR1I2 (0.50) CASRNR1I2ALDH1A1LMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010039913-A1 CALCILYTIC COMPOUNDS GLAXOSMITHKLINE LLC (US) 2010-04-08 WO disclosed