SCHEMBL28653100

SCHEMBL28653100

O=C(O)N1C[C@H]2C[C@H](NCc3ccccc3)C[C@H]2C1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DPP8 Q6V1X1 2/20 0.48
DPP9 Q86TI2 2/20 0.48
DPP7 Q9UHL4 2/20 0.48
ACHE P22303 5/20 0.46
BACE1 P56817 5/20 0.46
BCHE P06276 4/20 0.46
DRD4 P21917 1/20 0.45
DPP4 P27487 1/20 0.44
FYN P06241 1/20 0.44
GRIN2B Q13224 3/20 0.44
FABP6 P51161 1/20 0.43
ARG1 P05089 1/20 0.42
ARG2 P78540 1/20 0.42
MEN1 O00255 1/20 0.41
RAB9A P51151 1/20 0.41
KMT2A Q03164 1/20 0.41
KDM1A O60341 1/20 0.41
MAOA P21397 1/20 0.41
EPHX2 P34913 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11889380 1.00 DPP8 (0.48) DPP8DPP9DPP7ACHEBACE1
SCHEMBL11889561 1.00 DPP8 (0.48) DPP8DPP9DPP7ACHEBACE1
SCHEMBL11889448 0.90 DRD4 (0.49) DPP8DPP9DPP7ACHEBACE1
SCHEMBL11889388 0.90 DRD4 (0.49) DPP8DPP9DPP7ACHEBACE1
SCHEMBL20766109 0.87 BCHE (0.46) ACHEBACE1BCHEGRIN2BMEN1
SCHEMBL10320157 0.82 JAK1 (0.54) ACHEKMT2A
SCHEMBL22435955 0.82 JAK1 (0.54) ACHEKMT2A
SCHEMBL4875893 0.82 JAK1 (0.54) ACHEKMT2A
SCHEMBL10449417 0.82 JAK1 (0.54) ACHEKMT2A
SCHEMBL14699811 0.80 ACHE (0.49) ACHEBACE1BCHEFYNGRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113631557-A JAK kinase inhibitor, preparation method thereof and application thereof in medical field 上海华汇拓医药科技有限公司 2021-11-09 CN disclosed