SCHEMBL28655853

SCHEMBL28655853

C[Si](C)(C)CCOCn1ccc(Cl)c1-c1ccncn1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.36
MAP4K4 O95819 3/20 0.35
EGFR P00533 3/20 0.35
FRK P42685 3/20 0.35
MAPK9 P45984 3/20 0.35
SLK Q9H2G2 2/20 0.35
CSNK1D P48730 1/20 0.35
MAPT P10636 1/20 0.33
DGAT1 O75907 3/20 0.33
CSNK1A1 P48729 2/20 0.30
MAPK13 O15264 1/20 0.30
MAPK12 P53778 1/20 0.30
MAPK11 Q15759 1/20 0.30
MAPK14 Q16539 1/20 0.30
DCLK1 O15075 1/20 0.30
PRKD3 O94806 1/20 0.30
PRKACA P17612 1/20 0.30
FLT3 P36888 1/20 0.30
GSK3B P49841 1/20 0.30
MINK1 Q8N4C8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28672953 0.82 DGAT1 (0.36) MAPTDGAT1MAPK13MAPK12MAPK11
SCHEMBL29855368 0.77 MAPT (0.35) CYP2D6MAP4K4EGFRFRKMAPK9
SCHEMBL22613097 0.77 MAPT (0.35) CYP2D6MAP4K4EGFRFRKMAPK9
SCHEMBL30668712 0.76 MAP4K4 (0.39) CYP2D6MAP4K4EGFRFRKMAPK9
SCHEMBL20744175 0.76 MAP4K4 (0.39) CYP2D6MAP4K4EGFRFRKMAPK9
SCHEMBL28601695 0.72 DGAT1 (0.41) DGAT1
SCHEMBL1494550 0.70 DGAT1 (0.39) CYP2D6MAP4K4EGFRFRKMAPK9
SCHEMBL352030 0.69 FGFR1 (0.35) EGFRMAPTDGAT1FLT3
SCHEMBL30296433 0.69 DGAT1 (0.35) DGAT1
SCHEMBL29854726 0.69 FGFR1 (0.35) EGFRMAPTDGAT1FLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113727975-A Substituted pyrrolopyridines as JAK inhibitors 阿克拉瑞斯治疗股份有限公司 2021-11-30 CN disclosed