SCHEMBL28656529

SCHEMBL28656529

O=C(O)N1CCN2C(=O)c3cc(F)c(Br)cc3OC[C@H]2C1

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 1/20 0.37
KRAS P01116 10/20 0.34
AXL P30530 2/20 0.33
AKR1B1 P15121 1/20 0.32
TIPARP Q7Z3E1 5/20 0.31
PARP1 P09874 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
PARP12 Q9H0J9 1/20 0.30
PARP2 Q9UGN5 1/20 0.30
SOS1 Q07889 3/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26129936 0.89 GRIA1 (0.34) KRASAKR1B1TIPARPCYP2C9CYP2C19
SCHEMBL26108338 0.89 GRIA1 (0.34) KRASAKR1B1TIPARPCYP2C9CYP2C19
SCHEMBL28664244 0.87 KRAS (0.37) DPP4KRASAXLTIPARP
SCHEMBL23496870 0.87 KRAS (0.35) DPP4KRASAXLAKR1B1TIPARP
SCHEMBL23496692 0.87 KRAS (0.35) DPP4KRASAXLAKR1B1TIPARP
SCHEMBL24558178 0.84 USP30 (0.39) DPP4KRAS
SCHEMBL28658815 0.82 KRAS (0.41) DPP4KRAS
SCHEMBL26686750 0.81 DPP4 (0.36) DPP4KRASTIPARPPARP1CYP2C9
SCHEMBL23496779 0.80 KRAS (0.41) DPP4KRAS
SCHEMBL28654658 0.80 KRAS (0.40) DPP4KRAS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113508118-A Fused tricyclic compounds useful as anticancer agents 阿斯利康(瑞典)有限公司 2021-10-15 CN disclosed