SCHEMBL28656757

SCHEMBL28656757

O=C(O)c1ccc(-c2nc3ncc(Br)cc3[nH]2)cc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 1/20 0.64
MMP9 P14780 1/20 0.64
MMP8 P22894 1/20 0.64
MMP13 P45452 1/20 0.64
AURKA O14965 1/20 0.62
TBK1 Q9UHD2 6/20 0.55
IKBKE Q14164 5/20 0.55
DYRK1B Q9Y463 1/20 0.54
PTGDR2 Q9Y5Y4 2/20 0.53
HDAC6 Q9UBN7 1/20 0.51
ALDH1A1 P00352 2/20 0.50
KDM4E B2RXH2 2/20 0.50
KMT2A Q03164 2/20 0.50
HPGD P15428 1/20 0.50
MAPK10 P53779 1/20 0.49
DHODH Q02127 1/20 0.48
MEN1 O00255 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CHEK2 O96017 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4059275 0.88 AURKA (0.58) MMP2MMP9MMP8MMP13AURKA
SCHEMBL4148154 0.85 AURKA (0.52) MMP2MMP9MMP8MMP13AURKA
SCHEMBL1667430 0.83 AURKA (0.68) AURKADYRK1BPTGDR2ALDH1A1KMT2A
SCHEMBL4060567 0.80 AURKA (0.68) AURKAPTGDR2HDAC6ALDH1A1KDM4E
SCHEMBL18764092 0.79 HDAC6 (0.54) AURKATBK1IKBKEHDAC6ALDH1A1
Trifluoroacetic Acid SCHEMBL4843990 0.78 AURKA (0.56) MMP2MMP9MMP8MMP13AURKA
SCHEMBL4151626 0.77 AURKA (0.43) MMP2MMP9MMP8MMP13AURKA
SCHEMBL4053079 0.77 AURKA (0.67) AURKATBK1IKBKEDYRK1BALDH1A1
SCHEMBL14022277 0.76 PRMT5 (0.67) AURKAALDH1A1KDM4EKMT2AHPGD
SCHEMBL4054884 0.75 AURKA (0.61) AURKAPTGDR2HDAC6ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113544129-A Tricyclic compound preparation method and application thereof in medicine field 上海华汇拓医药科技有限公司 2021-10-22 CN disclosed