Glycine

Glycine

SCHEMBL28657486

NC(=O)c1ncc(-c2cccc(Cl)c2)cc1O.NCC(=O)O

nearest known ligand 0.65

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADORA1ADORA2AADORA2BADORA3PDE3APDE3BPDE4APDE4BPDE4CPDE4D

The experimentally established mechanism targets of Glycine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 14/20 0.65
EGLN3 Q9H6Z9 6/20 0.65
VEGFA P15692 5/20 0.65
FLT1 P17948 5/20 0.65
TET3 O43151 1/20 0.65
BBOX1 O75936 1/20 0.65
ASPH Q12797 1/20 0.65
TET2 Q6N021 1/20 0.65
KDM8 Q8N371 1/20 0.65
OGFOD1 Q8N543 1/20 0.65
TET1 Q8NFU7 1/20 0.65
HIF1AN Q9NWT6 1/20 0.65
IKBKB O14920 1/20 0.44
MAP4K4 O95819 1/20 0.44
GAA P10253 1/20 0.43
ALOX5 P09917 1/20 0.43
FTO Q9C0B1 1/20 0.42
GRIN1 Q05586 1/20 0.42
GRIN2B Q13224 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30346108 0.92 EGLN1 (0.63) EGLN1EGLN3VEGFAFLT1TET3
SCHEMBL3031409 0.92 EGLN1 (0.63) EGLN1EGLN3VEGFAFLT1TET3
Acetic Acid SCHEMBL23501731 0.90 EGLN1 (0.61) EGLN1EGLN3VEGFAFLT1TET3
Acetic Acid Methyl Ester SCHEMBL30471482 0.84 EGLN1 (0.64) EGLN1EGLN3VEGFAFLT1TET3
SCHEMBL4370919 0.83 EGLN1 (0.68) EGLN1EGLN3VEGFAFLT1TET3
SCHEMBL30514566 0.83 EGLN1 (0.68) EGLN1EGLN3VEGFAFLT1TET3
Vadadustat SCHEMBL29405970 0.79 EGLN1 (1.00) EGLN1EGLN3VEGFAFLT1TET3
Vadadustat SCHEMBL29357486 0.79 EGLN1 (1.00) EGLN1EGLN3VEGFAFLT1TET3
SCHEMBL1921394 0.79 EGLN1 (0.64) EGLN1EGLN3VEGFAFLT1TET3
Vadadustat SCHEMBL1920738 0.79 EGLN1 (1.00) EGLN1EGLN3VEGFAFLT1TET3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109593084-B Prolyl hydroxylase small-molecule photosensitive prodrug and preparation method and application thereof 中国药科大学 2021-09-28 CN disclosed