SCHEMBL28658271

SCHEMBL28658271

O=Cc1ccc(NCc2cccc(OC(F)(F)F)c2)nc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM5A P29375 1/20 0.50
KDM4C Q9H3R0 1/20 0.50
KDM5B Q9UGL1 1/20 0.50
HDAC1 Q13547 1/20 0.47
CCNT1 O60563 1/20 0.45
PIM1 P11309 2/20 0.45
P2RX7 Q99572 1/20 0.44
KCNN3 Q9UGI6 1/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
CHRM2 P08172 1/20 0.44
CHRM1 P11229 1/20 0.44
CHRM3 P20309 1/20 0.44
ALDH1A1 P00352 1/20 0.44
POLB P06746 1/20 0.44
ROCK1 Q13464 2/20 0.43
ROCK2 O75116 1/20 0.43
MAPK14 Q16539 1/20 0.43
ATM Q13315 1/20 0.43
GRM2 Q14416 1/20 0.42
ADORA3 P0DMS8 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28658424 0.86 KDM5A (0.53) KDM5AKDM4CKDM5BHDAC1P2RX7
SCHEMBL28925381 0.85 KDM5A (0.49) KDM5AKDM4CKDM5BCCNT1PIM1
SCHEMBL22102122 0.83 KDM5A (0.49) KDM5AKDM4CKDM5BCCNT1PIM1
SCHEMBL18525587 0.83 KDM5A (0.49) KDM5AKDM4CKDM5BCCNT1PIM1
SCHEMBL18525794 0.81 KDM5A (0.59) KDM5AKDM4CKDM5BPIM1ROCK1
SCHEMBL28658094 0.81 KDM5A (0.47) KDM5AKDM4CKDM5BCCNT1PIM1
SCHEMBL18525795 0.81 KDM5A (0.53) KDM5AKDM4CKDM5BPIM1L3MBTL1
SCHEMBL18526087 0.80 MAPK14 (0.53) KDM5AKDM4CKDM5BHDAC1CCNT1
SCHEMBL22102194 0.78 KDM5A (0.49) KDM5AKDM4CKDM5BCCNT1PIM1
SCHEMBL18526203 0.78 ROCK2 (0.56) KDM5AKDM4CKDM5BPIM1ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113412113-A Aminooxazine amides 豪夫迈·罗氏有限公司 2021-09-17 CN claimed
CN-113412113-A Aminooxazine amides 豪夫迈·罗氏有限公司 2021-09-17 CN disclosed