SCHEMBL28660932

SCHEMBL28660932

O=C1CC(c2cc(F)c(F)c(F)c2)CN1Cc1ccncc1Br

nearest known ligand 0.77

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.39
TSHR P16473 1/20 0.39
PDE10A Q9Y233 1/20 0.36
ALDH1A1 P00352 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
PDE4A P27815 3/20 0.34
PDE4B Q07343 3/20 0.34
PDE4C Q08493 3/20 0.34
PDE4D Q08499 3/20 0.34
PLA2G7 Q13093 1/20 0.32
DPP4 P27487 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29832754 1.00 HPGD (0.39) HPGDTSHRPDE10AALDH1A1SMN1; SMN2
SCHEMBL31030927 1.00 HPGD (0.39) HPGDTSHRPDE10AALDH1A1SMN1; SMN2
SCHEMBL28655573 0.90 HPGD (0.40) HPGDTSHRPDE10AALDH1A1SMN1; SMN2
SCHEMBL29832669 0.90 HPGD (0.40) HPGDTSHRPDE10AALDH1A1SMN1; SMN2
SCHEMBL20475363 0.90 HPGD (0.41) HPGDTSHRPDE10AALDH1A1SMN1; SMN2
SCHEMBL20475338 0.87 HPGD (0.41) HPGDTSHRPDE10AALDH1A1SMN1; SMN2
SCHEMBL31030949 0.87 HPGD (0.39) HPGDTSHRPDE10AALDH1A1SMN1; SMN2
App-311 SCHEMBL20475353 0.87 HPGD (0.39) HPGDTSHRPDE10AALDH1A1SMN1; SMN2
App-311 SCHEMBL31153157 0.87 HPGD (0.39) HPGDTSHRPDE10AALDH1A1SMN1; SMN2
SCHEMBL31030958 0.87 HPGD (0.39) HPGDTSHRPDE10AALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113549052-B 4-phenyl-1- (pyridine-4-ylmethyl) pyrrolidine-2-ketone derivative and preparation method and application thereof 首都医科大学脑重大疾病研究中心(北京脑重大疾病研究院) 2022-09-02 CN disclosed
CN-113549052-A 4-phenyl-1- (pyridine-4-ylmethyl) pyrrolidine-2-ketone derivative and preparation method and application thereof 首都医科大学脑重大疾病研究中心(北京脑重大疾病研究院) 2021-10-26 CN disclosed