SCHEMBL28662011

SCHEMBL28662011

COS(=O)(=O)CC1CCN(c2ccnc3ccccc23)CC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.49
NCF1 P14598 1/20 0.49
F10 P00742 2/20 0.46
KCNH2 Q12809 2/20 0.44
ALDH1A1 P00352 2/20 0.41
HTT P42858 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
KDM4E B2RXH2 1/20 0.41
GAA P10253 1/20 0.41
PKM P14618 1/20 0.41
PDGFRB P09619 1/20 0.41
DRD2 P14416 5/20 0.41
DRD3 P35462 3/20 0.41
NPC1 O15118 1/20 0.40
AKT1 P31749 1/20 0.39
HTR1A P08908 2/20 0.38
HTR2A P28223 2/20 0.38
HTR7 P34969 2/20 0.38
HTR6 P50406 2/20 0.38
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18980002 0.81 F10 (0.51) ADRB2NCF1F10KCNH2ALDH1A1
SCHEMBL29722200 0.81 F10 (0.51) ADRB2NCF1F10KCNH2ALDH1A1
SCHEMBL28250636 0.80 ADRB2 (0.50) ADRB2NCF1F10KCNH2ALDH1A1
SCHEMBL21034181 0.79 ADRB2 (0.49) ADRB2NCF1F10KCNH2ALDH1A1
SCHEMBL28438206 0.79 NPC1 (0.40) SMN1; SMN2NPC1
SCHEMBL28664473 0.79 ADRB2 (0.51) ADRB2NCF1F10KCNH2ALDH1A1
SCHEMBL24010608 0.78 ADRB2 (0.48) ADRB2NCF1F10KCNH2ALDH1A1
SCHEMBL6186822 0.77 ADRB2 (0.62) ADRB2NCF1F10KCNH2PDGFRB
SCHEMBL29722401 0.77 ADRB2 (0.58) ADRB2NCF1F10KCNH2ALDH1A1
SCHEMBL18980471 0.77 ADRB2 (0.58) ADRB2NCF1F10KCNH2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108699032-B Polycyclic TLR7/8 antagonists and their use in the treatment of immune disorders 默克专利有限公司 2022-07-22 CN disclosed
CN-113603675-A Polycyclic TLR7/8 antagonists and their use in the treatment of immune disorders 默克专利有限公司 2021-11-05 CN disclosed