SCHEMBL28665643

SCHEMBL28665643

O=C(O)N1CCN(C(=O)O)C(CN2C(=O)c3ccccc3C2=O)C1

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.45
SMN1; SMN2 Q16637 3/20 0.45
GAA P10253 3/20 0.45
MEN1 O00255 1/20 0.45
HSD17B10 Q99714 4/20 0.43
ALDH1A1 P00352 3/20 0.43
ALOX15 P16050 1/20 0.43
TSHR P16473 1/20 0.43
CA12 O43570 1/20 0.43
CA9 Q16790 1/20 0.43
MAPK1 P28482 1/20 0.43
HPGD P15428 1/20 0.41
KEAP1 Q14145 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15485406 0.85 KMT2A (0.48) KMT2ASMN1; SMN2GAAMEN1HSD17B10
SCHEMBL28688165 0.85 PARP1 (0.45) KMT2ASMN1; SMN2GAAMEN1HSD17B10
SCHEMBL20956786 0.81 HRH3 (0.48) HSD17B10ALDH1A1CA12CA9MAPK1
SCHEMBL5430075 0.81 HRH3 (0.48) HSD17B10ALDH1A1CA12CA9MAPK1
SCHEMBL23119906 0.78 CA12 (0.43) KMT2AMEN1ALDH1A1CA12CA9
SCHEMBL20956682 0.78 CA12 (0.43) KMT2AMEN1ALDH1A1CA12CA9
SCHEMBL21551126 0.77 KEAP1 (0.47) CA12CA9KEAP1
SCHEMBL23910438 0.77 SMN1; SMN2 (0.47) KMT2ASMN1; SMN2GAAMEN1ALDH1A1
SCHEMBL20479505 0.77 PARP1 (0.46) KMT2A
SCHEMBL17068112 0.77 PARP1 (0.46) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107922394-B 3-tetrazolyl-benzene-1, 2-disulfonamide derivatives as metallo-beta-lactamase inhibitors 默沙东公司 2021-07-13 CN disclosed