SCHEMBL28674012

SCHEMBL28674012

COC(=O)C(C)NC(=O)c1ccccn1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.55
ALDH1A1 P00352 3/20 0.55
HTT P42858 2/20 0.55
MEN1 O00255 1/20 0.53
KMT2A Q03164 1/20 0.53
APOBEC3G Q9HC16 1/20 0.53
SMN1; SMN2 Q16637 6/20 0.52
NPC1 O15118 3/20 0.52
RAB9A P51151 3/20 0.52
PKM P14618 2/20 0.52
MAPT P10636 1/20 0.52
GAA P10253 1/20 0.51
HPGD P15428 1/20 0.50
CDK5 Q00535 1/20 0.50
PAX8 Q06710 1/20 0.50
CDK5R1 Q15078 1/20 0.50
ALPL P05186 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
ACACB O00763 1/20 0.49
GRM4 Q14833 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4987029 0.86 SMN1; SMN2 (0.54) KDM4EALDH1A1HTTSMN1; SMN2NPC1
SCHEMBL1106971 0.85 KDM4E (0.63) KDM4EALDH1A1HTTSMN1; SMN2NPC1
SCHEMBL15549120 0.85 KDM4E (0.52) KDM4EALDH1A1HTTSMN1; SMN2NPC1
SCHEMBL15549121 0.85 KDM4E (0.52) KDM4EALDH1A1HTTSMN1; SMN2NPC1
SCHEMBL8580257 0.84 KDM4C (0.66) KDM4EALDH1A1HTTMEN1KMT2A
SCHEMBL8580260 0.84 KDM4C (0.66) KDM4EALDH1A1HTTMEN1KMT2A
SCHEMBL35210922 0.84 KDM4E (0.51) KDM4EALDH1A1HTTSMN1; SMN2NPC1
SCHEMBL28684226 0.83 ATM (0.57) KDM4EALDH1A1HTTSMN1; SMN2PKM
SCHEMBL27863520 0.83 KDM4E (0.56) KDM4EALDH1A1HTTSMN1; SMN2NPC1
SCHEMBL38655692 0.81 GAA (0.51) KDM4EALDH1A1HTTSMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114008053-A Prodrugs of NMDA receptor modulators H.隆德贝克有限公司 2022-02-01 CN disclosed