SCHEMBL286761

SCHEMBL286761

NC(=O)OC(Cl)c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.48
CYP1A2 P05177 1/20 0.48
PKM P14618 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
ALOX5 P09917 1/20 0.44
EPHX1 P07099 1/20 0.44
SRC P12931 1/20 0.41
TSHR P16473 1/20 0.41
LMNA P02545 3/20 0.40
MAPK1 P28482 2/20 0.40
CTSD P07339 1/20 0.39
KMT2A Q03164 1/20 0.39
SLC6A3 Q01959 3/20 0.39
DRD3 P35462 2/20 0.39
ADORA3 P0DMS8 1/20 0.39
EDNRB P24530 1/20 0.39
MC4R P32245 1/20 0.39
CYP2C19 P33261 1/20 0.39
MC3R P41968 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL984298 0.83 CYP2D6 (0.44) CYP2D6SRCTSHRLMNAMAPK1
SCHEMBL1096587 0.83 CYP2D6 (0.44) CYP2D6SRCTSHRLMNAMAPK1
SCHEMBL27840777 0.83 CYP2D6 (0.44) CYP2D6SRCTSHRLMNAMAPK1
SCHEMBL825537 0.81 CYP2D6 (0.48) CYP2D6SRCTSHRLMNAMAPK1
SCHEMBL1408551 0.79 ALDH1A1 (0.55) CYP2D6ALOX5SRCTSHRLMNA
SCHEMBL9815844 0.79 ESR1 (0.42) CYP2D6SRCTSHRLMNAMAPK1
SCHEMBL7464800 0.79 SMN1; SMN2 (0.44) CYP2D6CYP1A2PKMSMN1; SMN2NPSR1
SCHEMBL7454241 0.79 SMN1; SMN2 (0.44) CYP2D6CYP1A2PKMSMN1; SMN2NPSR1
SCHEMBL7454235 0.79 SMN1; SMN2 (0.44) CYP2D6CYP1A2PKMSMN1; SMN2NPSR1
SCHEMBL5306707 0.78 CYP2D6 (0.52) CYP2D6CYP1A2PKMSMN1; SMN2NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 675 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026089784-A2 COMPOUNDS AND COMPOSITIONS FOR CONJUGATION TO BIOLIGANDS FOR IMAGING AND RADIOPHARMACEUTICAL APPLICATIONS THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 2026-04-30 WO disclosed
WO-2025151874-A1 INDOLE ALKALOID ANTIPLASMODIAL AGENTS AND PREPARATION THEREOF UNIVERSITY OF CENTRAL FLORIDA RESEARCH FOUNDATION, INC. (US) 2025-07-17 WO disclosed
WO-2024147060-A1 NOVEL IONIZABLE LIPID COMPOUNDS FOR NUCLEIC ACID DELIVERY CELON PHARMA S.A. (PL) 2024-07-11 WO disclosed
WO-2024133853-A1 BIS-ESTER AND AMIDE CATIONIC LIPIDS SANOFI (FR) 2024-06-27 WO disclosed
WO-2024112854-A1 INHIBITORS OF RIPK2 AND MEDICAL USES THEREOF ODYSSEY THERAPEUTICS, INC. (US) 2024-05-30 WO disclosed
EP-4370132-A2 MULTIPLEXING TARGETING LIGANDS THROUGH CLICK CHEMISTRY AT THE ANOMERIC SITE OF SUGARS Alnylam Pharmaceuticals, Inc. (US) 2024-05-22 EP disclosed
EP-4370503-A1 ESTERS OF A RETINOID AND BAKUCHIOL AND PREPARATIONS THEREOF Conagen Inc. (US) 2024-05-22 EP disclosed
WO-2024097228-A1 COMPOUNDS TARGETING CDK11 AND METHODS OF USING THE SAME MELIORA THERAPEUTICS, INC. (US) 2024-05-10 WO disclosed
WO-2024097746-A1 ALKENE CYCLOPROPANATION WITH NICKEL CATALYST ENHANCER AND IMPROVED REARRANGEMENT REACTION CONAGEN INC. (US) 2024-05-10 WO disclosed
WO-2024086826-A2 POLYPEPTIDYL LINKERS Quantum-Si Incorporated (US) 2024-04-25 WO disclosed
WO-2005001047-A2 N-CARBOBENZYLOXY (N-CBZ)-DEPROTECTING ENZYME AND USES THEREFOR BRISTOL-MYERS SQUIBB COMPANY (US) 2005-01-06 WO disclosed
EP-1348025-A2 ENZYMATIC DEPROTECTION OF AMINES AND HYDROXIDES Bristol-Myers Squibb Company (US) 2003-10-01 EP disclosed
WO-2002053724-A2 ENZYMATIC DEPROTECTION OF AMINES AND HYDROXIDES BRISTOL-MYERS SQUIBB COMPANY (US) 2002-07-11 WO disclosed
CN-1311787-A oxazolidinone derivatives, process for their preparation and pharmaceutical compositions containing them ASTRA ZENECA CO LTD (SE) 2001-09-05 CN disclosed
CN-1284060-A Novel metalloprotease inhibitors FUJI YAKUHIN KOGYO KK (JP) 2001-02-14 CN disclosed
EP-0970066-A1 AMINOEPOXIDES FROM AMINOALDEHYDES AND IN-SITU FORMED HALOMETHYL ORGANOMETALLIC REAGENT G.D. SEARLE & CO. (US) 2000-01-12 EP disclosed
WO-1998029401-A1 AMINOEPOXIDES FROM AMINOALDEHYDES AND IN-SITU FORMED HALOMETHYL ORGANOMETALLIC REAGENT G.D. SEARLE & CO. (US) 1998-07-09 WO disclosed
EP-0804410-A1 METHOD OF PREPARING RETROVIRAL PROTEASE INHIBITOR INTERMEDIATES G.D. SEARLE & CO. (US) 1997-11-05 EP disclosed
EP-0730570-A1 METHOD FOR MAKING INTERMEDIATES USEFUL IN SYNTHESIS OF RETROVIRAL PROTEASE INHIBITORS G.D. SEARLE & CO. (US) 1996-09-11 EP disclosed
WO-1996022275-A1 METHOD OF PREPARING RETROVIRAL PROTEASE INHIBITOR INTERMEDIATES G.D. SEARLE & CO. (US) 1996-07-25 WO disclosed