SCHEMBL28680370

SCHEMBL28680370

CC(C)(C)OC(=O)NC(CCC(=O)OCc1ccccc1)C(=O)Nc1ccc(C(=O)O)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F10 P00742 1/20 0.48
PRSS1 P07477 1/20 0.48
CTSS P25774 2/20 0.48
CTSK P43235 1/20 0.48
SIRT1 Q96EB6 7/20 0.47
SIRT2 Q8IXJ6 7/20 0.47
HDAC4 P56524 2/20 0.47
HDAC1 Q13547 2/20 0.47
PPARA Q07869 2/20 0.47
PPARG P37231 1/20 0.47
HDAC8 Q9BY41 2/20 0.46
MEN1 O00255 1/20 0.46
ALDH1A1 P00352 1/20 0.46
HPGD P15428 1/20 0.46
KMT2A Q03164 1/20 0.46
SIRT5 Q9NXA8 1/20 0.46
HDAC3 O15379 1/20 0.46
HDAC7 Q8WUI4 1/20 0.46
HDAC2 Q92769 1/20 0.46
HDAC10 Q969S8 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30861278 0.93 SIRT2 (0.53) CTSSCTSKSIRT1SIRT2HDAC4
SCHEMBL2698182 0.93 SIRT2 (0.53) CTSSCTSKSIRT1SIRT2HDAC4
SCHEMBL28673197 0.90 KLK7 (0.53) CTSSCTSKSIRT1SIRT2HDAC4
SCHEMBL28673199 0.90 KLK7 (0.53) CTSSCTSKSIRT1SIRT2HDAC4
SCHEMBL20253483 0.89 HDAC8 (0.50) F10PRSS1CTSSCTSKSIRT1
SCHEMBL8431546 0.87 PPARA (0.55) CTSSCTSKPPARAPPARGMEN1
SCHEMBL8430542 0.87 PPARA (0.55) CTSSCTSKPPARAPPARGMEN1
SCHEMBL13359605 0.85 KMT2A (0.54) F10PRSS1SIRT1SIRT2HDAC4
SCHEMBL29361609 0.85 SIRT2 (0.58) CTSKSIRT1SIRT2HDAC4HDAC1
SCHEMBL14263348 0.84 MEN1 (0.54) SIRT1SIRT2HDAC8MEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113943259-A Amino acid derivative, preparation method and application thereof 西安禾渼生物医药有限公司 2022-01-18 CN disclosed