SCHEMBL28686167

SCHEMBL28686167

O=C(O)c1cccc(N2CC[C@@H](O)C2)c1Cl

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 9/20 0.55
TSHR P16473 1/20 0.44
PRKAB2 O43741 4/20 0.41
PRKAG1 P54619 4/20 0.41
PRKAA2 P54646 4/20 0.41
PRKAA1 Q13131 4/20 0.41
PRKAG3 Q9UGI9 4/20 0.41
PRKAG2 Q9UGJ0 4/20 0.41
PRKAB1 Q9Y478 4/20 0.41
ALDH1A1 P00352 1/20 0.39
P2RX7 Q99572 1/20 0.39
KMT2A Q03164 1/20 0.38
IRAK4 Q9NWZ3 1/20 0.38
PTPN1 P18031 1/20 0.37
AR P10275 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28697278 1.00 NOTUM (0.55) NOTUMTSHRPRKAB2PRKAG1PRKAA2
SCHEMBL29749785 0.92 NOTUM (0.49) NOTUMTSHRALDH1A1KMT2AIRAK4
SCHEMBL29627833 0.92 NOTUM (0.49) NOTUMTSHRALDH1A1KMT2AIRAK4
SCHEMBL29627850 0.91 NOTUM (0.50) NOTUMTSHRALDH1A1KMT2APTPN1
SCHEMBL28706635 0.91 NOTUM (0.48) NOTUMTSHRALDH1A1KMT2AIRAK4
SCHEMBL28686207 0.91 NOTUM (0.48) NOTUMTSHRALDH1A1KMT2AIRAK4
SCHEMBL28691758 0.90 NOTUM (0.49) NOTUMTSHRALDH1A1KMT2APTPN1
SCHEMBL29627823 0.88 TSHR (0.49) NOTUMTSHRALDH1A1
SCHEMBL28698733 0.87 TSHR (0.47) NOTUMTSHRALDH1A1
SCHEMBL29627843 0.82 TSHR (0.49) NOTUMTSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114072405-A Heterocyclic monoacylglycerol lipase (MAGL) inhibitors 豪夫迈·罗氏有限公司 2022-02-18 CN disclosed