SCHEMBL28689286

SCHEMBL28689286

COc1ccc2ncnc(N3CCC(C(C)CNS(N)(=O)=O)CC3)c2c1

nearest known ligand 0.72

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ENPP1 P22413 13/20 0.72
MTNR1B P49286 2/20 0.53
KIT P10721 1/20 0.46
PDGFRB P09619 1/20 0.45
USP2 O75604 3/20 0.43
CYP1A2 P05177 3/20 0.43
CYP3A4 P08684 3/20 0.43
CYP2C19 P33261 3/20 0.43
CLK4 Q9HAZ1 3/20 0.43
ALDH1A1 P00352 2/20 0.43
LMNA P02545 2/20 0.43
CYP2D6 P10635 2/20 0.43
MAPK1 P28482 2/20 0.43
HIF1A Q16665 2/20 0.43
HSD17B10 Q99714 1/20 0.42
MEN1 O00255 1/20 0.42
TSHR P16473 1/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31457627 1.00 ENPP1 (0.72) ENPP1MTNR1BKITPDGFRBUSP2
SCHEMBL28931602 0.93 ENPP1 (0.61) ENPP1MTNR1BKITPDGFRB
SCHEMBL22455020 0.87 ENPP1 (0.71) ENPP1MAPK1
SCHEMBL22441577 0.85 ENPP1 (0.52) ENPP1MTNR1BCYP3A4ALDH1A1LMNA
SCHEMBL28689284 0.85 ENPP1 (0.56) ENPP1MTNR1BKITPDGFRBUSP2
SCHEMBL20782514 0.84 ENPP1 (1.00) ENPP1MTNR1B
SCHEMBL22455035 0.83 ENPP1 (0.66) ENPP1PDGFRBMAPK1
SCHEMBL31457626 0.80 ENPP1 (0.48) ENPP1ALDH1A1MEN1KMT2A
SCHEMBL22441609 0.80 ENPP1 (0.48) ENPP1ALDH1A1MEN1KMT2A
SCHEMBL24391547 0.78 ENPP1 (0.82) ENPP1MTNR1BKITPDGFRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113924092-A Quinoline and quinazoline compounds and methods of use thereof 斯汀格瑞治疗股份有限公司 2022-01-11 CN disclosed