SCHEMBL28690649

SCHEMBL28690649

O=C(Nc1ccc(=O)n(-c2ccccc2)c1)C1CCCCC1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.60
PTPN1 P18031 1/20 0.52
ALDH1A1 P00352 3/20 0.52
GRM4 Q14833 1/20 0.52
TSHR P16473 2/20 0.49
KCNK3 O14649 1/20 0.49
KCNK9 Q9NPC2 1/20 0.49
ENPP3 O14638 3/20 0.48
ENPP1 P22413 3/20 0.48
ENPP2 Q13822 2/20 0.48
MEN1 O00255 1/20 0.48
GAA P10253 1/20 0.48
MAPT P10636 1/20 0.48
GFER P55789 1/20 0.48
KMT2A Q03164 1/20 0.48
HSD17B10 Q99714 2/20 0.47
KDM4E B2RXH2 1/20 0.47
NPC1 O15118 1/20 0.47
USP2 O75604 1/20 0.46
POLB P06746 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28700605 1.00 HPGD (0.60) HPGDPTPN1ALDH1A1GRM4TSHR
SCHEMBL28685818 0.99 HPGD (0.57) HPGDPTPN1ALDH1A1GRM4TSHR
SCHEMBL28704844 0.96 HPGD (0.54) HPGDPTPN1ALDH1A1GRM4TSHR
SCHEMBL28706297 0.93 KMT2A (0.55) HPGDPTPN1ALDH1A1TSHRMEN1
SCHEMBL28933271 0.82 EPHX2 (0.64) HPGDALDH1A1TSHRMEN1GFER
SCHEMBL28691401 0.81 EPHX2 (0.62) HPGDMEN1KMT2ANPC1SMN1; SMN2
SCHEMBL28691382 0.77 EPHX2 (0.54) HPGDALDH1A1GAAMAPTKMT2A
SCHEMBL19703413 0.76 HPGD (1.00) HPGDPTPN1ALDH1A1KCNK3KCNK9
SCHEMBL1300190 0.76 HPGD (1.00) HPGDPTPN1ALDH1A1KCNK3KCNK9
SCHEMBL21653300 0.75 PTPN1 (0.54) HPGDPTPN1ALDH1A1ENPP3ENPP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114057630-B Pirfenidone derivative and synthetic method and application thereof 郑州大学 2023-06-02 CN claimed
CN-114057630-A Pirfenidone derivative and synthetic method and application thereof 郑州大学 2022-02-18 CN claimed
CN-114057630-B Pirfenidone derivative and synthetic method and application thereof 郑州大学 2023-06-02 CN disclosed
CN-114057630-A Pirfenidone derivative and synthetic method and application thereof 郑州大学 2022-02-18 CN disclosed