SCHEMBL28690986

SCHEMBL28690986

Cc1ccc(CN(C)c2cnc(-c3ccccc3)c(-c3ccccc3)n2)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CKS1B P61024 2/20 0.59
SKP1 P63208 2/20 0.59
SKP2 Q13309 2/20 0.59
CNR1 P21554 5/20 0.57
MAPT P10636 3/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
TSHR P16473 1/20 0.47
KMT2A Q03164 1/20 0.47
TDP1 Q9NUW8 2/20 0.44
CYP19A1 P11511 1/20 0.41
LMNA P02545 3/20 0.40
KDM4E B2RXH2 3/20 0.40
HTT P42858 1/20 0.40
ALDH1A1 P00352 3/20 0.40
NPC1 O15118 1/20 0.40
HPGD P15428 1/20 0.40
RAB9A P51151 1/20 0.40
ESR1 P03372 1/20 0.39
ESR2 Q92731 1/20 0.39
TP53 P04637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30725791 1.00 CKS1B (0.59) CKS1BSKP1SKP2CNR1MAPT
SCHEMBL30725783 0.96 CNR1 (0.62) CKS1BSKP1SKP2CNR1MAPT
SCHEMBL28707155 0.96 CNR1 (0.62) CKS1BSKP1SKP2CNR1MAPT
SCHEMBL28691774 0.88 CKS1B (0.57) CKS1BSKP1SKP2CNR1MAPT
SCHEMBL30725764 0.88 CKS1B (0.57) CKS1BSKP1SKP2CNR1MAPT
SCHEMBL28691799 0.88 CKS1B (0.57) CKS1BSKP1SKP2CNR1MAPT
SCHEMBL30725778 0.88 CKS1B (0.57) CKS1BSKP1SKP2CNR1MAPT
SCHEMBL30725763 0.85 CKS1B (0.55) CKS1BSKP1SKP2CNR1MAPT
SCHEMBL28697301 0.85 CKS1B (0.55) CKS1BSKP1SKP2CNR1MAPT
SCHEMBL30725780 0.85 CKS1B (0.57) CKS1BSKP1SKP2CNR1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118206499-A 2,3, 5-Trisubstituted pyrazine compound and preparation method and application thereof 郑州大学 2024-06-18 CN disclosed
CN-118146165-A 2,3, 5-Trisubstituted pyrazine compound and preparation method and application thereof 郑州大学 2024-06-07 CN disclosed
CN-113968824-B 2,3, 5-trisubstituted pyrazine compound and preparation method and application thereof 郑州大学 2024-01-19 CN disclosed
CN-113968824-A 2,3, 5-trisubstituted pyrazine compound and preparation method and application thereof 郑州大学 2022-01-25 CN disclosed