SCHEMBL28697301

SCHEMBL28697301

CN(Cc1ccc(C(C)(C)C)cc1)c1cnc(-c2ccccc2)c(-c2ccccc2)n1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CKS1B P61024 2/20 0.55
SKP1 P63208 2/20 0.55
SKP2 Q13309 2/20 0.55
CYP19A1 P11511 2/20 0.44
CNR1 P21554 1/20 0.43
MAPT P10636 3/20 0.41
KMT2A Q03164 3/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
TSHR P16473 1/20 0.41
TP53 P04637 1/20 0.41
MEN1 O00255 2/20 0.41
RAB9A P51151 1/20 0.41
NR1I2 O75469 2/20 0.40
KCNH2 Q12809 2/20 0.40
LMNA P02545 1/20 0.40
ADRA2A P08913 1/20 0.40
CYP2D6 P10635 1/20 0.40
ACHE P22303 1/20 0.40
SLC6A2 P23975 1/20 0.40
HTR2A P28223 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30725763 1.00 CKS1B (0.55) CKS1BSKP1SKP2CYP19A1CNR1
SCHEMBL28690986 0.85 CKS1B (0.59) CKS1BSKP1SKP2CYP19A1CNR1
SCHEMBL30725791 0.85 CKS1B (0.59) CKS1BSKP1SKP2CYP19A1CNR1
SCHEMBL30725778 0.84 CKS1B (0.57) CKS1BSKP1SKP2CNR1MAPT
SCHEMBL30725764 0.84 CKS1B (0.57) CKS1BSKP1SKP2CYP19A1CNR1
SCHEMBL28691774 0.84 CKS1B (0.57) CKS1BSKP1SKP2CNR1MAPT
SCHEMBL28691799 0.84 CKS1B (0.57) CKS1BSKP1SKP2CYP19A1CNR1
SCHEMBL30725777 0.82 CKS1B (0.55) CKS1BSKP1SKP2CYP19A1CNR1
SCHEMBL30725783 0.82 CNR1 (0.62) CKS1BSKP1SKP2CYP19A1CNR1
SCHEMBL28707155 0.82 CNR1 (0.62) CKS1BSKP1SKP2CYP19A1CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118206499-A 2,3, 5-Trisubstituted pyrazine compound and preparation method and application thereof 郑州大学 2024-06-18 CN disclosed
CN-118146165-A 2,3, 5-Trisubstituted pyrazine compound and preparation method and application thereof 郑州大学 2024-06-07 CN disclosed
CN-113968824-B 2,3, 5-trisubstituted pyrazine compound and preparation method and application thereof 郑州大学 2024-01-19 CN disclosed
CN-113968824-A 2,3, 5-trisubstituted pyrazine compound and preparation method and application thereof 郑州大学 2022-01-25 CN disclosed