SCHEMBL28696221

SCHEMBL28696221

Oc1ccc(-c2cc(OCC3CNC3)c3cn[nH]c3c2)nc1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TDO2 P48775 2/20 0.36
JAK2 O60674 7/20 0.36
JAK1 P23458 7/20 0.36
TYK2 P29597 7/20 0.36
JAK3 P52333 7/20 0.36
PIM1 P11309 6/20 0.35
PIK3CD O00329 4/20 0.35
GSK3B P49841 3/20 0.35
PIK3CA P42336 2/20 0.35
PIK3CB P42338 2/20 0.35
KDM1A O60341 1/20 0.33
FGFR1 P11362 1/20 0.33
FGFR2 P21802 1/20 0.33
FGFR3 P22607 1/20 0.33
PIK3CG P48736 2/20 0.32
SGK1 O00141 1/20 0.32
IRAK4 Q9NWZ3 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL28681300 0.92 PIM1 (0.35) TDO2JAK2JAK1TYK2JAK3
SCHEMBL30161646 0.88 PIK3CD (0.47) TDO2JAK2JAK1TYK2JAK3
SCHEMBL20699367 0.88 PIK3CD (0.47) TDO2JAK2JAK1TYK2JAK3
SCHEMBL28681297 0.83 CYP4F2 (0.33) TDO2PIM1SGK1IRAK4
SCHEMBL28931797 0.82 JAK3 (0.51) TDO2JAK2JAK1TYK2JAK3
SCHEMBL28689643 0.82 FGFR1 (0.48) TDO2JAK2JAK1TYK2JAK3
Trifluoroacetic Acid SCHEMBL29608317 0.80 PIK3CD (0.45) TDO2JAK2JAK1TYK2JAK3
Trifluoroacetic Acid SCHEMBL28680413 0.80 PIK3CD (0.45) TDO2JAK2JAK1TYK2JAK3
SCHEMBL20699380 0.80 PIM1 (0.46) TDO2JAK2JAK1TYK2JAK3
SCHEMBL20699377 0.80 PIM1 (0.46) TDO2JAK2JAK1TYK2JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113831326-A Condensed heterocyclic derivative and application thereof in medicine 四川海思科制药有限公司 2021-12-24 CN disclosed