SCHEMBL28689643

SCHEMBL28689643

Oc1ccc(-c2cc(OCC3CNC3)c3cn[nH]c3c2)c(F)c1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 3/20 0.48
FGFR2 P21802 2/20 0.48
HASPIN Q8TF76 1/20 0.39
JAK2 O60674 9/20 0.38
JAK1 P23458 9/20 0.38
TYK2 P29597 9/20 0.38
JAK3 P52333 9/20 0.38
PIM1 P11309 1/20 0.36
KCNH2 Q12809 1/20 0.36
PIM2 Q9P1W9 1/20 0.36
SGK1 O00141 1/20 0.36
USP7 Q93009 1/20 0.35
TDO2 P48775 1/20 0.34
PIK3CD O00329 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
HDAC5 Q9UQL6 1/20 0.34
ESR1 P03372 1/20 0.34
ESR2 Q92731 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL28687582 0.93 FGFR1 (0.42) FGFR1FGFR2HASPINJAK2JAK1
SCHEMBL28931797 0.88 JAK3 (0.51) FGFR1FGFR2JAK2JAK1TYK2
SCHEMBL20699367 0.85 PIK3CD (0.47) FGFR1FGFR2JAK2JAK1TYK2
SCHEMBL30161646 0.85 PIK3CD (0.47) FGFR1FGFR2JAK2JAK1TYK2
Trifluoroacetic Acid SCHEMBL28686997 0.82 JAK3 (0.47) FGFR1JAK2JAK1TYK2JAK3
SCHEMBL20699403 0.82 JAK3 (0.49) FGFR1FGFR2JAK2JAK1TYK2
SCHEMBL30161719 0.82 JAK3 (0.49) FGFR1FGFR2JAK2JAK1TYK2
SCHEMBL28696221 0.82 TDO2 (0.36) FGFR1FGFR2JAK2JAK1TYK2
SCHEMBL28672841 0.82 FGFR1 (0.41) FGFR1FGFR2HASPINJAK2JAK1
SCHEMBL28687763 0.81 JAK3 (0.57) JAK2JAK1TYK2JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113831326-A Condensed heterocyclic derivative and application thereof in medicine 四川海思科制药有限公司 2021-12-24 CN disclosed