SCHEMBL28696572

SCHEMBL28696572

N[C@H](CCCC(O)c1cc(F)c(F)cc1F)CC(=O)O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR2 O95136 1/20 0.38
S1PR1 P21453 1/20 0.38
CYP3A4 P08684 3/20 0.37
ADRA2A P08913 2/20 0.37
ADRA2B P18089 2/20 0.37
ADRA2C P18825 2/20 0.37
ADRA1A P35348 2/20 0.37
ADRB2 P07550 1/20 0.37
HSD17B10 Q99714 1/20 0.37
KDM4E B2RXH2 1/20 0.36
MAPT P10636 1/20 0.36
APEX1 P27695 1/20 0.36
RAD52 P43351 1/20 0.36
RECQL P46063 1/20 0.36
BLM P54132 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
KDM4C Q9H3R0 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
DPP4 P27487 4/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28033030 0.77 ADRA2A (0.39) CYP3A4ADRA2AADRA2BADRA2CADRA1A
SCHEMBL25417892 0.77 DPP4 (0.42) S1PR2S1PR1CYP3A4DPP4
SCHEMBL27912553 0.77 DPP4 (0.42) S1PR2S1PR1CYP3A4DPP4
SCHEMBL28183873 0.77 DPP4 (0.42) S1PR2S1PR1CYP3A4DPP4
SCHEMBL28183878 0.76 S1PR2 (0.43) S1PR2S1PR1CYP3A4DPP4
SCHEMBL26107941 0.73 DPP4 (0.44) S1PR2S1PR1CYP3A4DPP4
SCHEMBL27916012 0.73 DPP4 (0.44) S1PR2S1PR1CYP3A4DPP4
SCHEMBL25415095 0.73 DPP4 (0.44) S1PR2S1PR1CYP3A4DPP4
SCHEMBL744345 0.70 DPP4 (0.39) DPP4FFAR1
SCHEMBL12971465 0.70 DPP4 (0.39) DPP4FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107286164-B Application of compound in preparation of sitagliptin and method for preparing sitagliptin 武汉臻智生物科技有限公司 2021-08-03 CN disclosed