SCHEMBL28697606

SCHEMBL28697606

C#CCN(Cc1ccc(C(=O)NO)cc1)Cc1ccccc1C

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 13/20 0.52
HDAC8 Q9BY41 6/20 0.52
HDAC1 Q13547 14/20 0.47
HDAC3 O15379 2/20 0.46
HDAC7 Q8WUI4 2/20 0.46
HDAC10 Q969S8 2/20 0.46
PYCR1 P32322 2/20 0.43
HDAC2 Q92769 2/20 0.43
RORC P51449 1/20 0.41
HDAC4 P56524 1/20 0.41
HDAC11 Q96DB2 1/20 0.41
HDAC9 Q9UKV0 1/20 0.41
HDAC5 Q9UQL6 1/20 0.41
KDM4E B2RXH2 1/20 0.41
LMNA P02545 1/20 0.41
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28673090 0.87 HDAC6 (0.50) HDAC6HDAC8HDAC1HDAC3HDAC7
SCHEMBL28690762 0.86 HDAC1 (0.61) HDAC6HDAC8HDAC1HDAC3HDAC7
SCHEMBL28697601 0.86 HDAC6 (0.53) HDAC6HDAC8HDAC1HDAC3HDAC7
SCHEMBL28691803 0.85 HDAC1 (0.55) HDAC6HDAC8HDAC1HDAC3HDAC2
SCHEMBL28696676 0.85 HDAC6 (0.60) HDAC6HDAC8HDAC1HDAC3HDAC7
SCHEMBL28700013 0.84 HDAC1 (0.54) HDAC6HDAC8HDAC1HDAC3HDAC7
SCHEMBL28688145 0.81 HDAC6 (0.52) HDAC6HDAC8HDAC1HDAC3HDAC7
SCHEMBL28697641 0.80 HDAC6 (0.56) HDAC6HDAC8HDAC1HDAC3HDAC7
SCHEMBL28690802 0.80 HDAC6 (0.56) HDAC6HDAC8HDAC1HDAC3HDAC7
SCHEMBL28699833 0.79 CA1 (0.59) HDAC6HDAC8HDAC1PYCR1HDAC11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113956182-B HDAC/MAO-B dual inhibitor and preparation and application thereof 杭州师范大学 2023-11-17 CN disclosed
CN-113956182-A HDAC/MAO-B dual inhibitor and preparation and application thereof 杭州师范大学 2022-01-21 CN disclosed