SCHEMBL28697641

SCHEMBL28697641

C#CCN(Cc1ccc(F)cc1)Cc1ccc(C(=O)NO)cc1

nearest known ligand 0.56

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 16/20 0.56
HDAC8 Q9BY41 13/20 0.56
HDAC11 Q96DB2 4/20 0.54
HDAC3 O15379 6/20 0.50
PYCR1 P32322 4/20 0.50
HDAC1 Q13547 4/20 0.48
HDAC7 Q8WUI4 1/20 0.46
HDAC10 Q969S8 1/20 0.46
NCOR2 Q9Y618 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28674189 0.87 HDAC6 (0.55) HDAC6HDAC8HDAC11HDAC3PYCR1
SCHEMBL28690762 0.87 HDAC1 (0.61) HDAC6HDAC8HDAC11HDAC3PYCR1
SCHEMBL28690802 0.86 HDAC6 (0.56) HDAC6HDAC8HDAC3PYCR1HDAC1
SCHEMBL28696676 0.86 HDAC6 (0.60) HDAC6HDAC8HDAC11HDAC3PYCR1
SCHEMBL28697601 0.85 HDAC6 (0.53) HDAC6HDAC8HDAC11HDAC3PYCR1
SCHEMBL28699833 0.83 CA1 (0.59) HDAC6HDAC8HDAC11PYCR1HDAC1
SCHEMBL28696678 0.82 HDAC6 (0.52) HDAC6HDAC8HDAC11HDAC3PYCR1
SCHEMBL28696862 0.82 HDAC6 (0.51) HDAC6HDAC8HDAC3PYCR1HDAC1
SCHEMBL28673090 0.81 HDAC6 (0.50) HDAC6HDAC8HDAC3PYCR1HDAC1
SCHEMBL28697606 0.80 HDAC6 (0.52) HDAC6HDAC8HDAC11HDAC3PYCR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113956182-A HDAC/MAO-B dual inhibitor and preparation and application thereof 杭州师范大学 2022-01-21 CN disclosed