SCHEMBL28697971

SCHEMBL28697971

CCOC(=O)c1nnn(-c2ccc(OCOC)c(F)c2)c1C

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.57
ALOX12 P18054 1/20 0.57
MAPT P10636 2/20 0.54
SMN1; SMN2 Q16637 2/20 0.47
KMT2A Q03164 1/20 0.46
ALDH1A1 P00352 4/20 0.44
SLC5A1 P13866 3/20 0.44
SLC5A2 P31639 3/20 0.44
MITF O75030 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
HPGD P15428 1/20 0.43
SPR P35270 1/20 0.43
PTGS2 P35354 1/20 0.43
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA4 P22748 1/20 0.42
CA9 Q16790 1/20 0.42
MET P08581 1/20 0.42
NPC1 O15118 1/20 0.41
LMNA P02545 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29408091 1.00 TP53 (0.57) TP53ALOX12MAPTSMN1; SMN2KMT2A
SCHEMBL28686848 0.87 TP53 (0.57) TP53ALOX12MAPTSMN1; SMN2KMT2A
SCHEMBL29408088 0.87 TP53 (0.57) TP53ALOX12MAPTSMN1; SMN2KMT2A
SCHEMBL3400622 0.85 TP53 (0.66) TP53ALOX12MAPTSMN1; SMN2KMT2A
SCHEMBL29408102 0.81 NOTUM (0.51) TP53MAPTALDH1A1PTGS2MET
SCHEMBL28685562 0.81 NOTUM (0.51) TP53MAPTALDH1A1PTGS2MET
SCHEMBL29408101 0.81 NOTUM (0.51) TP53MAPTALDH1A1PTGS2MET
SCHEMBL3406655 0.80 POLB (0.62) TP53ALOX12MAPTSMN1; SMN2KMT2A
SCHEMBL28697962 0.79 KCNN4 (0.36) TP53MAPTKMT2AALDH1A1HPGD
SCHEMBL29408072 0.79 KCNN4 (0.36) TP53MAPTKMT2AALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114127066-A Inhibitors of indoleamine 2, 3-dioxygenase and/or tryptophan 2, 3-dioxygenase 爱杜西亚药品有限公司 2022-03-01 CN disclosed