SCHEMBL29408102

SCHEMBL29408102

COCOc1ccc(-n2nnc(CO)c2C)cc1F

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.51
GRIN1 Q05586 10/20 0.43
GRIN2B Q13224 10/20 0.43
RXRA P19793 10/20 0.42
KCNN4 O15554 1/20 0.40
MET P08581 2/20 0.35
CYP1A2 P05177 1/20 0.35
GAA P10253 1/20 0.34
TP53 P04637 1/20 0.34
MAPT P10636 1/20 0.34
PTGS2 P35354 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29408101 1.00 NOTUM (0.51) NOTUMGRIN1GRIN2BRXRAKCNN4
SCHEMBL28685562 1.00 NOTUM (0.51) NOTUMGRIN1GRIN2BRXRAKCNN4
SCHEMBL28685629 0.85 NOTUM (0.58) NOTUMGRIN1GRIN2BRXRAGAA
SCHEMBL29408092 0.85 NOTUM (0.58) NOTUMGRIN1GRIN2BRXRAGAA
SCHEMBL28697962 0.81 KCNN4 (0.36) GRIN1GRIN2BRXRAKCNN4MET
SCHEMBL29408072 0.81 KCNN4 (0.36) GRIN1GRIN2BRXRAKCNN4MET
SCHEMBL29408091 0.81 TP53 (0.57) METTP53MAPTPTGS2ALDH1A1
SCHEMBL28697971 0.81 TP53 (0.57) METTP53MAPTPTGS2ALDH1A1
SCHEMBL19232450 0.74 GRIN1 (0.64) NOTUMGRIN1GRIN2BRXRA
SCHEMBL22684398 0.74 NOTUM (0.63) NOTUMGRIN1GRIN2BRXRACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114127066-A Inhibitors of indoleamine 2, 3-dioxygenase and/or tryptophan 2, 3-dioxygenase 爱杜西亚药品有限公司 2022-03-01 CN disclosed