SCHEMBL28699149

SCHEMBL28699149

CC(C)(C)OC(=O)N1CCN(c2ccc3c(c2)CN(C(=O)OCc2ccccc2)C3)CC1

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TMEM97 Q5BJF2 20/20 0.77
SIGMAR1 Q99720 20/20 0.77
HRH1 P35367 6/20 0.77
HRH3 Q9Y5N1 6/20 0.77
HRH2 P25021 5/20 0.77
HTR1A P08908 3/20 0.77
ADRA2A P08913 3/20 0.77
ADRA2B P18089 3/20 0.77
HTR2C P28335 3/20 0.77
ADRA2C P18825 2/20 0.77
HTR1E P28566 2/20 0.77
HTR2A P28223 2/20 0.77
HTR2B P41595 2/20 0.77
DRD1 P21728 1/20 0.77
HTR1B P28222 1/20 0.77
SLC6A4 P31645 1/20 0.77
ADRB1 P08588 1/20 0.68
CHRM1 P11229 1/20 0.65
SLC6A2 P23975 1/20 0.65
DRD3 P35462 2/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30449380 1.00 TMEM97 (0.77) TMEM97SIGMAR1HRH1HRH3HRH2
SCHEMBL5456675 0.90 TMEM97 (0.70) TMEM97SIGMAR1HRH1HRH3HRH2
SCHEMBL19521478 0.87 TMEM97 (1.00) TMEM97SIGMAR1HRH1HRH3HRH2
SCHEMBL21800330 0.86 TMEM97 (0.60) TMEM97SIGMAR1HRH1HRH3HRH2
SCHEMBL23673943 0.85 TMEM97 (0.56) TMEM97SIGMAR1HRH1HRH3HRH2
SCHEMBL29974284 0.85 TMEM97 (0.56) TMEM97SIGMAR1HRH1HRH3HRH2
SCHEMBL22529537 0.85 TMEM97 (0.56) TMEM97SIGMAR1HRH1HRH3HRH2
SCHEMBL21591628 0.84 TMEM97 (0.60) TMEM97SIGMAR1HRH1HRH3HRH2
SCHEMBL23854670 0.84 TMEM97 (0.60) TMEM97SIGMAR1HRH1HRH3HRH2
SCHEMBL21800260 0.84 TMEM97 (0.57) TMEM97SIGMAR1HRH1HRH3HRH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114075219-B Quinoline condensed ring derivative, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2023-11-14 CN disclosed
CN-114621230-B Nitrogen-containing heterocyclic compound, preparation method thereof and application thereof in medicine 江苏恒瑞医药股份有限公司 2023-06-16 CN disclosed
CN-114276351-B Nitrogen-containing heterocyclic derivative, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2023-06-16 CN disclosed
CN-114621230-A Nitrogen-containing heterocyclic compound, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2022-06-14 CN disclosed
CN-114276351-A Nitrogenous heterocyclic derivative, preparation method thereof and application thereof in medicine 江苏恒瑞医药股份有限公司 2022-04-05 CN disclosed
CN-114075219-A Quinoline condensed ring derivative, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2022-02-22 CN disclosed